Efficient synthesis of substituted biaryl anilines and biaryl phenols via a Suzuki cross-coupling reaction

被引：23

作者：

Liu, B ^{[1
]}

Moffett, KK ^{[1
]}

Joseph, RW ^{[1
]}

Dorsey, BD ^{[1
]}

机构：

[1] Locus Pharmaceut Inc, Blue Bell, PA 19422 USA

来源：

TETRAHEDRON LETTERS | 2005年 / 46卷 / 11期

关键词：

Suzuki coupling; Pd catalyst; biaryl building blocks;

D O I：

10.1016/j.tetlet.2005.01.125

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient synthesis of biaryl building blocks with multiple point diversities via a Suzuki cross-coupling reaction using a commercially available preformed Pd catalyst 1 was reported. Substituted biaryl anilines and phenols were obtained in one step from commercially available aryl halides. (C) 2005 Elsevier Ltd. All rights reserved.

引用

页码：1779 / 1782

页数：4

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