BIARYL SYNTHESIS VIA SUZUKI COUPLING ON A SOLID SUPPORT

被引：160
|
作者：
FRENETTE, R [1 ]
FRIESEN, RW [1 ]
机构：
[1] MERCK FROSST CTR THERAPEUT RES,DEPT MED CHEM,POINTE CLAIRE H9R 4P8,PQ,CANADA
来源：
TETRAHEDRON LETTERS | 1994年 / 35卷 / 49期
关键词：
D O I：
10.1016/0040-4039(94)88458-7
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Aryl boronic acids undergo a facile and efficient palladium catalyzed cross-coupling reaction with aryl bromides and iodides that are bound to a Merrifield resin. Simple transesterification releases the biaryl products from the solid support in excellent purity and yield.
引用
收藏
页码：9177 / 9180
页数：4
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