BIARYL SYNTHESIS VIA SUZUKI COUPLING ON A SOLID SUPPORT

被引：160
|
作者：
FRENETTE, R [1 ]
FRIESEN, RW [1 ]
机构：
[1] MERCK FROSST CTR THERAPEUT RES,DEPT MED CHEM,POINTE CLAIRE H9R 4P8,PQ,CANADA
来源：
TETRAHEDRON LETTERS | 1994年 / 35卷 / 49期
关键词：
D O I：
10.1016/0040-4039(94)88458-7
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Aryl boronic acids undergo a facile and efficient palladium catalyzed cross-coupling reaction with aryl bromides and iodides that are bound to a Merrifield resin. Simple transesterification releases the biaryl products from the solid support in excellent purity and yield.
引用
收藏
页码：9177 / 9180
页数：4
相关论文
共 50 条
  • [31] Synthesis of Ferrocenyl Porphyrins via Suzuki Coupling and Their Photophysical Properties
    Bakar, Muntaz A.
    Sergeeva, Natalia N.
    Juillard, Thomas
    Senge, Mathias O.
    [J]. ORGANOMETALLICS, 2011, 30 (11) : 3225 - 3228
  • [32] Efficient synthesis of isoflavone analogues via a Suzuki coupling reaction
    Ding, K
    Wang, SM
    [J]. TETRAHEDRON LETTERS, 2005, 46 (21) : 3707 - 3709
  • [33] An expedient synthesis of ellipticine via Suzuki-Miyaura coupling
    Konakahara, Takeo
    Kiran, Y. B.
    Okuno, Yuri
    Ikeda, Reiko
    Sakai, Norio
    [J]. TETRAHEDRON LETTERS, 2010, 51 (17) : 2335 - 2338
  • [34] New asymmetric synthesis of several biaryl diacids and dinaphthol via biaryl coupling reaction induced by chiral auxiliaries
    Qin, C
    Liu, M
    Song, LK
    Rong, GB
    [J]. CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2002, 22 (12) : 1013 - 1017
  • [35] SYNTHESIS OF NIGRICANIN VIA INTRAMOLECULAR BIARYL COUPLING REACTION OF FUNCTIONALIZED PHENYL BENZOATE
    Matsukihira, Takuya
    Kida, Tatsuya
    Hidaka, Kei
    Saga, Shumpei
    Takemura, Mami
    Yonoki, Atsuro
    Nishimori, Tsuyoshi
    Horino, Yoshikazu
    Harayama, Takashi
    Takeuchi, Yasuo
    Abe, Hitoshi
    [J]. HETEROCYCLES, 2013, 87 (12) : 2555 - 2565
  • [36] Suzuki-Miyaura Carbonylative Reaction in the Synthesis of Biaryl Ketones
    Zhu Zhuangli
    Zhang Weiqiang
    Gao Ziwei
    [J]. PROGRESS IN CHEMISTRY, 2016, 28 (11) : 1626 - 1633
  • [37] First total synthesis of tenuifolin via PIFA mediated oxidative biaryl coupling
    Tang, Changhua
    Li, Ziyuan
    Wang, Yiyun
    Xu, Jinyi
    Kong, Lingyi
    Yao, Hequan
    Wu, Xiaoming
    [J]. TETRAHEDRON LETTERS, 2011, 52 (26) : 3275 - 3278
  • [38] Solution-phase synthesis of an aminomethyl-substituted biaryl library via sequential amine N-alkylation and Suzuki cross-coupling
    Organ, MG
    Arvanitis, EA
    Dixon, CE
    Lavorato, DJ
    [J]. JOURNAL OF COMBINATORIAL CHEMISTRY, 2001, 3 (05): : 473 - 476
  • [39] Palladium nanoparticle catalysis: borylation of aryl and benzyl halides and one-pot biaryl synthesis via sequential borylation-Suzuki-Miyaura coupling
    Bej, Ansuman
    Srimani, Dipankar
    Sarkar, Amitabha
    [J]. GREEN CHEMISTRY, 2012, 14 (03) : 661 - 667
  • [40] Asymmetric Suzuki-Miyaura Cross-Coupling for the Synthesis of Chiral Biaryl Compounds as Potential Monophosphine Ligands
    Ma, Yan-Na
    Yang, Shang-Dong
    [J]. CHEMISTRY-A EUROPEAN JOURNAL, 2015, 21 (18) : 6673 - 6677
12345