Efficient synthesis of substituted biaryl anilines and biaryl phenols via a Suzuki cross-coupling reaction

被引：23
|
作者：
Liu, B [1 ]
Moffett, KK [1 ]
Joseph, RW [1 ]
Dorsey, BD [1 ]
机构：
[1] Locus Pharmaceut Inc, Blue Bell, PA 19422 USA
来源：
TETRAHEDRON LETTERS | 2005年 / 46卷 / 11期
关键词：
Suzuki coupling; Pd catalyst; biaryl building blocks;
D O I：
10.1016/j.tetlet.2005.01.125
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient synthesis of biaryl building blocks with multiple point diversities via a Suzuki cross-coupling reaction using a commercially available preformed Pd catalyst 1 was reported. Substituted biaryl anilines and phenols were obtained in one step from commercially available aryl halides. (C) 2005 Elsevier Ltd. All rights reserved.
引用
收藏
页码：1779 / 1782
页数：4
相关论文
共 50 条
  • [31] An efficient synthesis of 4-substituted coumarin derivatives via a palladium-catalyzed Suzuki cross-coupling reaction
    Rajale, Trideep
    Sharma, Shikha
    Stroud, Daniel A.
    Unruh, Daniel K.
    Miaou, Emily
    Lai, Kimberly
    Birney, David M.
    [J]. TETRAHEDRON LETTERS, 2014, 55 (49) : 6627 - 6630
  • [32] Efficient synthesis of functionalized 6-substituted-thiosalicylates via microwave-promoted Suzuki cross-coupling reaction
    Liu, Yu-Chao
    Qu, Ren-Yu
    Chen, Qiong
    Wu, Qiong-You
    Yang, Guang-Fu
    [J]. TETRAHEDRON, 2014, 70 (17) : 2746 - 2752
  • [33] Biaryl-substituted beta-lactam synthons via the Suzuki reaction.
    Bose, AK
    Rumthao, S
    Bhagavath, S
    Balasubramanian, KK
    Manhas, MS
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 223 : B141 - B141
  • [34] A biaryl cross-coupling strategy for functionalisation of benzocrown ethers
    Dixon, Sally
    Brown, Richard C. D.
    Gale, Philip A.
    [J]. CHEMICAL COMMUNICATIONS, 2007, (34) : 3565 - 3567
  • [35] The palladium catalysed biaryl cross-coupling of pyridazine triflates
    Aldous, DJ
    Bower, S
    Moorcroft, N
    Todd, M
    [J]. SYNLETT, 2001, (01) : 150 - 152
  • [36] SET-Induced Biaryl Cross-Coupling: An SRN1 Reaction
    Haines, Brandon E.
    Wiest, Olaf
    [J]. JOURNAL OF ORGANIC CHEMISTRY, 2014, 79 (06): : 2771 - 2774
  • [37] Suzuki coupling of diaryl tellurides for the synthesis of unsymmetrical biaryl compounds
    Jin, Jin
    Lolla, Mahati
    Zhang, Shaozhong
    Yen, Changchi
    Whippie, Drew
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251
  • [38] Synthesis of biaryl cyclic peptides through solid-phase borylation and cyclization by a Suzuki-Miyaura cross-coupling
    Afonso, A.
    Feliu, L.
    Planas, M.
    [J]. JOURNAL OF PEPTIDE SCIENCE, 2010, 16 : 48 - 48
  • [39] Facile preparation of novel β-substituted metalloporphyrins via Suzuki cross-coupling reaction
    Gauler, R
    Keuper, R
    Winter, A
    Risch, N
    [J]. ARKIVOC, 2004, : 48 - 56
  • [40] New asymmetric synthesis of several biaryl diacids and dinaphthol via biaryl coupling reaction induced by chiral auxiliaries
    Qin, C
    Liu, M
    Song, LK
    Rong, GB
    [J]. CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2002, 22 (12) : 1013 - 1017
12345