Copper-catalyzed three-component reaction of imidazo[1,2-a]pyridine with elemental sulfur and arylboronic acid to produce sulfenylimidazo[1,2-a]pyridines

被引:0
|
作者
Genhua Xiao [1 ]
Hao Min [1 ]
Zhilei Zheng [1 ]
Guobo Deng [1 ]
Yun Liang [1 ]
机构
[1] National & Local Joint Engineering Laboratory for New Petro-chemical Materials and Fine Utilization of Resources, Key Laboratory of Chemical Biology and Traditional Chinese Medicine Research, Ministry of Education, Key Laboratory of the Assembly and Applic
基金
中国国家自然科学基金;
关键词
Copper; Three-component; Pyridine; Sulfur; Arylboronic acids;
D O I
暂无
中图分类号
O626 [杂环化合物];
学科分类号
070303 ; 081704 ;
摘要
In this work, an efficient copper-catalyzed three-component reaction for the synthesis of sulfenylimidazo[1,2-a]pyridines using elemental sulfur as the sulfenylating agents has been developed. The reaction could proceed smoothly with a high degree of functional group tolerance and provide the desired products in moderate to good yield.
引用
收藏
页码:1363 / 1366
页数:4
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