Copper-catalyzed three-component reaction of imidazo[1,2-a]pyridine with elemental sulfur and arylboronic acid to produce sulfenylimidazo[1,2-a]pyridines

被引：0

作者：

Genhua Xiao ^{[1
]}

Hao Min ^{[1
]}

Zhilei Zheng ^{[1
]}

Guobo Deng ^{[1
]}

Yun Liang ^{[1
]}

机构：

[1] National & Local Joint Engineering Laboratory for New Petro-chemical Materials and Fine Utilization of Resources, Key Laboratory of Chemical Biology and Traditional Chinese Medicine Research, Ministry of Education, Key Laboratory of the Assembly and Applic

来源：

Chinese Chemical Letters | 2018年 / 29卷 / 09期

基金：

中国国家自然科学基金;

关键词：

Copper; Three-component; Pyridine; Sulfur; Arylboronic acids;

D O I：

暂无

中图分类号：

O626 [杂环化合物];

学科分类号：

070303 ; 081704 ;

摘要：

In this work, an efficient copper-catalyzed three-component reaction for the synthesis of sulfenylimidazo[1,2-a]pyridines using elemental sulfur as the sulfenylating agents has been developed. The reaction could proceed smoothly with a high degree of functional group tolerance and provide the desired products in moderate to good yield.

引用

页码：1363 / 1366

页数：4

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