CYCLOCONDENSATION OF N-(2-BROMOETHYL)PHTHALIMIDE WITH THE DIANION OF ISOBUTYRIC ACID TO A FUNCTIONALIZED 2,3-DIHYDROOXAZOLO[2,3]ISOINDOL-5(9BH)-ONE DERIVATIVE

被引：0

作者：

DEKIMPE, N ^{[1
]}

VIRAG, M ^{[1
]}

KEPPENS, M ^{[1
]}

SCHEINMANN, F ^{[1
]}

STACHULSKI, AV ^{[1
]}

机构：

[1] SALFORD ULTRAFINE CHEM & RES LTD,MANCHESTER M15 6SY,LANCS,ENGLAND

来源：

JOURNAL OF CHEMICAL RESEARCH-S | 1995年 / 06期

关键词：

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Contrary to a previous report describing that the condensation or N-(2-bromoethyl)phthalimide with the dianion of isobutyric acid affords 3-{2-[(aziridin-1-yl)carbonyl]phenyl}-2,2-dimethyl-3-oxopropanoic acid, we report that this reaction in fact leads to 2-(5-oxo-2,3,5,9b-tetrahydrooxazolo[2,3-a]isoindol-9b-yl)-2-methylpropanoic acid.

引用

页码：252 / 253

页数：2

共 41 条

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