A tandem Petasis-Ugi multi component condensation reaction: solution phase synthesis of six dimensional libraries

被引：56
|
作者：
Portlock, DE
Ostaszewski, R
Naskar, D
West, L
机构：
[1] Procter & Gamble Pharmaceut Hlth Care Res Ctr, Combinatorial Chem Sect, Mason, OH 45040 USA
[2] Warsaw Univ Technol, PL-00664 Warsaw, Poland
[3] Chembiotek Res Int, Salt Lake City 700091, Calcutta, India
来源：
TETRAHEDRON LETTERS | 2003年 / 44卷 / 03期
关键词：
D O I：
10.1016/S0040-4039(02)02619-9
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Amino acids with three points of diversity generated from the Petasis boronic acid-Mannich reaction can be used as one of the four components of the Ugi condensation to prepare six dimensional libraries of dipeptide amides. (C) 2002 Published by Elsevier Science Ltd.
引用
收藏
页码：603 / 605
页数：3
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