Synthesis of new 4-aryl/alkyl-1-(5′,5′-diphenyl-4′-oxo-1′-H-4′,5′-dihydroimidazolidin-2′-yl)-3-hydroxy-1,2,4-triazolidine-5-thione derivatives as potential anti-cancer agents

被引：0

作者：

Datar, PA ^{[1
]}

Shirodkar, PY ^{[1
]}

Panikkar, KR ^{[1
]}

机构：

[1] KM Kundnani Coll Pharm, Bombay 400018, Maharashtra, India

来源：

INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2003年 / 42卷 / 03期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

New 4-aryl/alkyl-1-(5',5'-diphenyl-4'-oxo- 1'H-4',5'-dihydroimidazolidin-2'-yl)-3-hydroxy-1,2,4-triazolidine-5-thiones 3 have been prepared by the reaction of 2-carbethoxy-(5',5'-diphenyl-4'-oxo-1'-H-4',5'-dihydroimidazolidin-2'-yl)-hydrazine 2 with various aryl/alkylisothiocyanates. Their anti-bacterial, anti-fungal, anthelmintic and anti-cancer activities are reported.

引用

页码：690 / 694

页数：5

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