An efficient synthesis of N-protected β-aminoethanesulfonyl chlorides:: Versatile building blocks for the synthesis of oligopeptidosulfonamides

被引：1
|
作者：
Brouwer, AJ [1 ]
Monnee, MCF [1 ]
Liskamp, RMJ [1 ]
机构：
[1] Univ Utrecht, Utrecht Inst Pharmaceut Sci, Dept Med Chem, NL-3508 TB Utrecht, Netherlands
来源：
SYNTHESIS-STUTTGART | 2000年 / 11期
关键词：
sulfonamides; sulfonyl chloride; amino acid; thioacetate; oxidation;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A very efficient method for the synthesis of beta-amino-ethanesulfonyl chlorides is described. These aliphatic functionalized sulfonyl chlorides are accessible starting from st variety of protected amino acids, including those having functionalized side chains.
引用
收藏
页码：1579 / 1584
页数：6
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