An efficient synthesis of N-protected β-aminoethanesulfonyl chlorides:: Versatile building blocks for the synthesis of oligopeptidosulfonamides

被引：1

作者：

Brouwer, AJ ^{[1
]}

Monnee, MCF ^{[1
]}

Liskamp, RMJ ^{[1
]}

机构：

[1] Univ Utrecht, Utrecht Inst Pharmaceut Sci, Dept Med Chem, NL-3508 TB Utrecht, Netherlands

来源：

SYNTHESIS-STUTTGART | 2000年 / 11期

关键词：

sulfonamides; sulfonyl chloride; amino acid; thioacetate; oxidation;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A very efficient method for the synthesis of beta-amino-ethanesulfonyl chlorides is described. These aliphatic functionalized sulfonyl chlorides are accessible starting from st variety of protected amino acids, including those having functionalized side chains.

引用

页码：1579 / 1584

页数：6

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