An efficient synthesis of N-protected β-aminoethanesulfonyl chlorides:: Versatile building blocks for the synthesis of oligopeptidosulfonamides

被引：1

作者：

Brouwer, AJ ^{[1
]}

Monnee, MCF ^{[1
]}

Liskamp, RMJ ^{[1
]}

机构：

[1] Univ Utrecht, Utrecht Inst Pharmaceut Sci, Dept Med Chem, NL-3508 TB Utrecht, Netherlands

来源：

SYNTHESIS-STUTTGART | 2000年 / 11期

关键词：

sulfonamides; sulfonyl chloride; amino acid; thioacetate; oxidation;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A very efficient method for the synthesis of beta-amino-ethanesulfonyl chlorides is described. These aliphatic functionalized sulfonyl chlorides are accessible starting from st variety of protected amino acids, including those having functionalized side chains.

引用

页码：1579 / 1584

页数：6

共 50 条

[1] Synthesis of N-phthalimido β-aminoethanesulfonyl chlorides:: the use of thionyl chloride for a simple and efficient synthesis of new peptidosulfonamide building blocks
Humljan, J
Gobec, S
TETRAHEDRON LETTERS, 2005, 46 (23) : 4069 - 4072
[2] Synthesis of N-protected staurosporinones
Wada, Yasuhiro
Nagasaki, Hideo
Tokuda, Masao
Orito, Kazuhiko
JOURNAL OF ORGANIC CHEMISTRY, 2007, 72 (06): : 2008 - 2014
[3] SYNTHESIS OF N-PROTECTED OXYTOCEINES
PHOTAKI, I
EXPERIENTIA, 1964, 20 (09): : 487 - &
[4] Synthesis of N-protected galactosamine building blocks from D-tagatose via the Heyns rearrangement
Wrodnigg, TM
Lundt, I
Stütz, AE
JOURNAL OF CARBOHYDRATE CHEMISTRY, 2006, 25 (01) : 33 - 41
[5] Synthesis of N-protected cyano aziridines
Fioravanti, S
Morreale, A
Pellacani, L
Tardella, PA
SYNLETT, 2004, (06) : 1083 - 1085
[6] A SIMPLE AND EFFICIENT SYNTHESIS OF N-PROTECTED IMIDAZOLE-4-CARBALDEHYDE
WINTER, J
RETEY, J
SYNTHESIS-STUTTGART, 1994, (03): : 245 - 246
[7] Synthesis of alkyl and aryl esthrs of N-protected β-homoamino acids from N-protected α-aminodiazoketones
Vasanthakumar, GR
Gopi, HN
Babu, VVS
PROTEIN AND PEPTIDE LETTERS, 2002, 9 (06): : 529 - 532
[8] SYNTHESIS OF N-PROTECTED ERYTHRO-PHENYLALANYLEPOXIDES
HEINSOO, A
RAIDARU, G
LINASK, K
JARV, J
ZETTERSTROM, M
LANGEL, U
TETRAHEDRON-ASYMMETRY, 1995, 6 (09) : 2245 - 2247
[9] Efficient synthesis of protected sulfonopeptides from N-protected 2-aminoalkyl xanthates and thioacetates
Kakaei, Saeed
Xu, Jiaxi
TETRAHEDRON, 2013, 69 (43) : 9068 - 9075
[10] Synthesis of N-protected azaoligosaccharides and their cyclic derivatives
Sawada, D
Takahashi, H
Shiro, M
Ikegami, S
TETRAHEDRON LETTERS, 2005, 46 (14) : 2399 - 2403

← 1 2 3 4 5 →