SYNTHESIS AND CHARACTERIZATION OF NOVEL PYRIMIDINE DERIVATIVES FROM 2,3-FURANDIONES

被引：4

作者：

Koca, Irfan ^{[1
]}

Yildirim, Ismail ^{[2
]}

机构：

[1] Bozok Univ, Fac Arts & Sci, Dept Chem, TR-66200 Yozgat, Turkey

[2] Erciyes Univ, Fac Arts & Sci, Dept Chem, TR-38039 Kayseri, Turkey

来源：

HETEROCYCLIC COMMUNICATIONS | 2009年 / 15卷 / 05期

关键词：

2,3-Furandione; pyrimidine-2(1H)-one; pyrimidine-2(1-H)-thione; nucleophilic cycloaddition; FUNCTIONALIZED; 1H-PYRIMIDINES; OXALYL COMPOUNDS; ENAMINONES; INHIBITORS; AGENTS; ACID;

D O I：

10.1515/HC.2009.15.5.377

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Various novel pyrimidine-2(1H)-one and pyrimidine-2(1H)-thione derivatives 3a-m have been synthesized efficiently in good yields by the treatment of 4-p-methylbenzoyl-5-p-methylphenyl-2,3-furandione (1a) and 4-(3,4-dimethoxybenzoyl)-5-(3,4-dimethoxyphenyl)-2,3-furandione (1b) with some ureas and thioureas 2. Structures of these compounds 3 were established on the basis of elemental analysis, IR, H-1- and C-13-NMR spectral studies.

引用

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页码：377 / 384

页数：8

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