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- [31] Oncogenic KRAS G12C: Kinetic and redox characterization of covalent inhibitionJOURNAL OF BIOLOGICAL CHEMISTRY, 2022, 298 (08)Huynh, Minh, V论文数: 0 引用数: 0 h-index: 0机构: Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USAParsonage, Derek论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Sch Med, Dept Biochem, Winston Salem, NC 27101 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USAForshaw, Tom E.论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Sch Med, Dept Internal Med, Sect Mol Med, Winston Salem, NC 27101 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USAChirasani, Venkat R.论文数: 0 引用数: 0 h-index: 0机构: Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USAHobbs, G. Aaron论文数: 0 引用数: 0 h-index: 0机构: Univ N Carolina, Dept Pharmacol, Chapel Hill, NC 27515 USA Univ N Carolina, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27515 USA Med Univ South Carolina, Charleston, SC 29425 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USAWu, Hanzhi论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Sch Med, Dept Internal Med, Sect Mol Med, Winston Salem, NC 27101 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USALee, Jingyun论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Baptist Comprehens Canc Ctr, Winston Salem, NC 27157 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USAFurdui, Cristina M.论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Sch Med, Dept Internal Med, Sect Mol Med, Winston Salem, NC 27101 USA Wake Forest Baptist Comprehens Canc Ctr, Winston Salem, NC 27157 USA Wake Forest Sch Med, Ctr Redox Biol & Med, Winston Salem, NC 27101 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USAPoole, Leslie B.论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Sch Med, Dept Biochem, Winston Salem, NC 27101 USA Wake Forest Baptist Comprehens Canc Ctr, Winston Salem, NC 27157 USA Wake Forest Sch Med, Ctr Redox Biol & Med, Winston Salem, NC 27101 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USACampbell, Sharon L.论文数: 0 引用数: 0 h-index: 0机构: Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USA Univ N Carolina, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27515 USA Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC 27515 USA
- [32] SRC kinase drives multidrug resistance induced by KRAS-G12C inhibitionSCIENCE ADVANCES, 2024, 10 (50):Song, Xinxin论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USAZhou, Zhuan论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USAElmezayen, Ammar论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Dept Biochem & Radiat Oncol, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USAWu, Runliu论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USAYu, Chunhua论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USAGao, Boning论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Hamon Ctr Therapeut Oncol Res, Harold C Simmons Comprehens Canc Ctr, Dept Pharmacol,Dept Internal Med, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USAMinna, John D.论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Hamon Ctr Therapeut Oncol Res, Harold C Simmons Comprehens Canc Ctr, Dept Pharmacol,Dept Internal Med, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USAWestover, Kenneth D.论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Dept Biochem & Radiat Oncol, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USAZeh, Herbert J.论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USA论文数: 引用数: h-index:机构:Heasley, Lynn E.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USA Rocky Mt Reg VA Med Ctr, Eastern Colorado VA Healthcare Syst, Aurora, CO 80045 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USAKang, Rui论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USATang, Daolin论文数: 0 引用数: 0 h-index: 0机构: UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USA UT Southwestern Med Ctr, Dept Surg, Dallas, TX 75390 USA
- [33] KRAS G12C mutated lung adenocarcinomas: a morphological and molecular cartographyVIRCHOWS ARCHIV, 2021, 479 : S162 - S162Pirlog, R.论文数: 0 引用数: 0 h-index: 0机构: UMF Iuliu Hatieganu, Cluj Napoca, Romania UMF Iuliu Hatieganu, Cluj Napoca, RomaniaPiton, N.论文数: 0 引用数: 0 h-index: 0机构: UMF Iuliu Hatieganu, Cluj Napoca, Romania UMF Iuliu Hatieganu, Cluj Napoca, RomaniaMarguet, F.论文数: 0 引用数: 0 h-index: 0机构: UMF Iuliu Hatieganu, Cluj Napoca, Romania UMF Iuliu Hatieganu, Cluj Napoca, RomaniaLamy, A.论文数: 0 引用数: 0 h-index: 0机构: UMF Iuliu Hatieganu, Cluj Napoca, Romania UMF Iuliu Hatieganu, Cluj Napoca, RomaniaSabourin, J.论文数: 0 引用数: 0 h-index: 0机构: UMF Iuliu Hatieganu, Cluj Napoca, Romania UMF Iuliu Hatieganu, Cluj Napoca, Romania
- [34] Combination of tipifarnib with KRAS G12C inhibitors to prevent adaptive resistanceCANCER RESEARCH, 2023, 83 (07)Patel, Hetika Vora论文数: 0 引用数: 0 h-index: 0Smith, Alison论文数: 0 引用数: 0 h-index: 0Chan, Stacia论文数: 0 引用数: 0 h-index: 0Kessler, Linda论文数: 0 引用数: 0 h-index: 0Burrows, Francis论文数: 0 引用数: 0 h-index: 0Malik, Shivani论文数: 0 引用数: 0 h-index: 0
- [35] Resistance looms for KRAS G12C inhibitors and rational tackling strategiesPHARMACOLOGY & THERAPEUTICS, 2022, 229Zhang, Junmin论文数: 0 引用数: 0 h-index: 0机构: Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R China Lanzhou Univ, Coll Chem & Chem Engn, State Key Lab Appl Organ Chem, Sch Pharm, Lanzhou 730000, Peoples R China Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R ChinaZhang, Juanhong论文数: 0 引用数: 0 h-index: 0机构: Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R China Lanzhou Univ, Coll Chem & Chem Engn, State Key Lab Appl Organ Chem, Sch Pharm, Lanzhou 730000, Peoples R China Northwest Normal Univ, Coll Life Sci, Lanzhou 730070, Peoples R China Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R ChinaLiu, Qing论文数: 0 引用数: 0 h-index: 0机构: Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R China Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R ChinaFan, Xing-Xing论文数: 0 引用数: 0 h-index: 0机构: Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R China Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R ChinaLeung, Elaine Lai-Han论文数: 0 引用数: 0 h-index: 0机构: Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R China Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R ChinaYao, Xiao-Jun论文数: 0 引用数: 0 h-index: 0机构: Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R China Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R ChinaLiu, Liang论文数: 0 引用数: 0 h-index: 0机构: Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R China Macau Univ Sci & Technol, Dr Nehes Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa, Macau Sar, Peoples R China
- [36] AXL signal mediates adaptive resistance to KRAS G12C inhibitors in KRAS G12C-mutant tumor cellsCANCER LETTERS, 2024, 587论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Hirai, Soichi论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanKatayama, Yuki论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanFukui, Sarina论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanSawada, Ryo论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanTachibana, Yusuke论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Ishida, Masaki论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan论文数: 引用数: h-index:机构:Kunimasa, Kei论文数: 0 引用数: 0 h-index: 0机构: Osaka Int Canc Inst, Dept Thorac Oncol, Osaka, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanSasaki, Takaaki论文数: 0 引用数: 0 h-index: 0机构: Asahikawa Med Univ, Dept Internal Med 1, Asahikawa, Hokkaido, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanNishida, Makoto论文数: 0 引用数: 0 h-index: 0机构: St Marianna Univ, Sch Med, Dept Internal Med, Div Resp Med, Kawasaki, Kanagawa, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanFuruya, Naoki论文数: 0 引用数: 0 h-index: 0机构: St Marianna Univ, Sch Med, Dept Internal Med, Div Resp Med, Kawasaki, Kanagawa, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanWatanabe, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Niigata Univ, Grad Sch Med & Dent Sci, Dept Resp Med & Infect Dis, Niigata, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanShiotsu, Shinsuke论文数: 0 引用数: 0 h-index: 0机构: Japanese Red Cross Kyoto Daiichi Hosp, Dept Resp Med, Kyoto, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanNishioka, Naoya论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan Fukuchiyama City Hosp, Dept Resp Med, Kyoto, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanHorinaka, Mano论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Drug Discovery Med, Kyoto, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanSakai, Toshiyuki论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Drug Discovery Med, Kyoto, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanUehara, Hisanori论文数: 0 引用数: 0 h-index: 0机构: Tokushima Univ Hosp, Div Pathol, Tokushima, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanYano, Seiji论文数: 0 引用数: 0 h-index: 0机构: Kanazawa Univ, Grad Sch Med Sci, Dept Resp Med, Kanazawa, Japan Kanazawa Univ, Canc Res Inst, Div Med Oncol, Kanazawa, Japan Kanazawa Univ, WPI Nano Life Sci Inst WPI Nano LSI, Kanazawa, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanSon, Bo-Kyung论文数: 0 引用数: 0 h-index: 0机构: Univ Tokyo, Inst Future Initiat, Tokyo, Japan Univ Tokyo, Inst Gerontol, Tokyo, Japan Univ Tokyo, Grad Sch Med, Dept Geriatr Med, Tokyo, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanTokuda, Shinsaku论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, JapanTakayama, Koichi论文数: 0 引用数: 0 h-index: 0机构: Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan Kyoto Prefectural Univ Med, Grad Sch Med Sci, Dept Pulm Med, 465,Kajii Cho,Kamigyo Ku, Kyoto 6028566, Japan
- [37] Concomitant KRAS mutations attenuate sensitivity of non-small cell lung cancer cells to KRAS G12C inhibitionScientific Reports, 12Tereza Vaclova论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyAtanu Chakraborty论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyJames Sherwood论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologySarah Ross论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyDanielle Carroll论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyJ. Carl Barrett论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyJulian Downward论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyElza C. de Bruin论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, Oncology
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- [39] KRAS G12C mutation is not undruggable anymoreBULLETIN DU CANCER, 2020, 107 (02) : 145 - 145Rodrigues, Manuel论文数: 0 引用数: 0 h-index: 0机构: INSERM, U830, Equipe Labellisee Ligue Natl Canc, DNA Repair & Uveal Melanoma DRUM, 26 Rue Ulm, F-75005 Paris, France PSL Res Univ, Inst Curie, Dept Oncol Med, F-75005 Paris, France INSERM, U830, Equipe Labellisee Ligue Natl Canc, DNA Repair & Uveal Melanoma DRUM, 26 Rue Ulm, F-75005 Paris, France
- [40] Concomitant KRAS mutations attenuate sensitivity of non-small cell lung cancer cells to KRAS G12C inhibitionSCIENTIFIC REPORTS, 2022, 12 (01)Vaclova, Tereza论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandChakraborty, Atanu论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Biosci, Cambridge CB2 0RE, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandSherwood, James论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut, Precis Med & Biosamples, Cambridge CB4 0WG, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandRoss, Sarah论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Biosci, Cambridge CB2 0RE, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandCarroll, Danielle论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandBarrett, J. Carl论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Translat Med, Waltham, MA 02451 USA AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England论文数: 引用数: h-index:机构:de Bruin, Elza C.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England