An improved synthesis of solid-supported reagents (SSRs) for selective acylation of amines by microwave irradiation

被引：26
|
作者：
Petricci, E [1 ]
Botta, M [1 ]
Corelli, F [1 ]
Mugnaini, C [1 ]
机构：
[1] Univ Studi Siena, Dipartimento Farm Chim Tecnol, I-53100 Siena, Italy
来源：
TETRAHEDRON LETTERS | 2002年 / 43卷 / 37期
关键词：
D O I：
10.1016/S0040-4039(02)01478-8
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Microwave-assisted acylation of a solid-Supported pyrimidine linker with different acyl chlorides gave polymer-bound 4-acyloxypyrimidines, which in turn were used as SSRs for rapid and selective acylation of amines under microwave irradiation. (C) 2002 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：6507 / 6509
页数：3
相关论文
共 50 条
  • [1] New solid-supported reagents (SSRs) for selective acylation of amines
    Botta, M
    Corelli, F
    Petricci, E
    Seri, C
    HETEROCYCLES, 2002, 56 (1-2) : 369 - 377
  • [2] Microwave-assisted acylation of amines, alcohols, and phenols by the use of solid-supported reagents (SSRs)
    Petricci, E
    Mugnaini, C
    Radi, M
    Corelli, F
    Botta, M
    JOURNAL OF ORGANIC CHEMISTRY, 2004, 69 (23): : 7880 - 7887
  • [3] Solid-supported Reagents in Organic Synthesis Using Microwave Irradiation
    Heravi, Majid M.
    Moghimi, Setareh
    CURRENT ORGANIC CHEMISTRY, 2013, 17 (05) : 504 - 527
  • [4] Solid-supported reagents in organic synthesis using microwave irradiation
    Department of Chemistry, School of Science, Alzahra University, PO Box 1993891176, Vanak, Tehran, Iran
    Heravi, M. M. (mmh1331@yahoo.com), 1600, Bentham Science Publishers (17):
  • [5] Solid-supported reagents in organic synthesis
    Drewry, DH
    Coe, DM
    Poon, S
    MEDICINAL RESEARCH REVIEWS, 1999, 19 (02) : 97 - 148
  • [6] Two efficient N-acylation methods mediated by solid-supported reagents for weakly nucleophilic heterocyclic amines
    Kim, K
    Le, K
    SYNLETT, 1999, (12) : 1957 - 1959
  • [7] A one-port, two-step microwave-assisted synthesis of highly functionalized benzoxazoles using solid-supported reagents (SSRs)
    Radi, Marco
    Saletti, Sara
    Botta, Maurizio
    TETRAHEDRON LETTERS, 2008, 49 (29-30) : 4464 - 4466
  • [8] Solid-supported tert-alkoxycarbonylation reagents for anchoring of amines during solid phase organic synthesis
    Hernandez, AS
    Hodges, JC
    JOURNAL OF ORGANIC CHEMISTRY, 1997, 62 (10): : 3153 - 3157
  • [9] Solid-Supported tert-Alkoxycarbonylation Reagents for Anchoring of Amines during Solid Phase Organic Synthesis
    Hernandez, A. S.
    Hodges, J. C.
    Journal of Organic Chemistry, 62 (10):
  • [10] Solid-supported Robinson annulation under microwave irradiation
    Takatori, K
    Nakayama, M
    Futaishi, N
    Yamada, S
    Hirayama, S
    Kajiwara, M
    CHEMICAL & PHARMACEUTICAL BULLETIN, 2003, 51 (04) : 455 - 457
12345