An improved synthesis of solid-supported reagents (SSRs) for selective acylation of amines by microwave irradiation

被引：26
|
作者：
Petricci, E [1 ]
Botta, M [1 ]
Corelli, F [1 ]
Mugnaini, C [1 ]
机构：
[1] Univ Studi Siena, Dipartimento Farm Chim Tecnol, I-53100 Siena, Italy
来源：
TETRAHEDRON LETTERS | 2002年 / 43卷 / 37期
关键词：
D O I：
10.1016/S0040-4039(02)01478-8
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Microwave-assisted acylation of a solid-Supported pyrimidine linker with different acyl chlorides gave polymer-bound 4-acyloxypyrimidines, which in turn were used as SSRs for rapid and selective acylation of amines under microwave irradiation. (C) 2002 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：6507 / 6509
页数：3
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