Microwave-assisted acylation of amines, alcohols, and phenols by the use of solid-supported reagents (SSRs)

被引：37
|
作者：
Petricci, E [1 ]
Mugnaini, C [1 ]
Radi, M [1 ]
Corelli, F [1 ]
Botta, M [1 ]
机构：
[1] Univ Siena, Dipartimento Farmaco Chim Tecnol, I-53100 Siena, Italy
来源：
JOURNAL OF ORGANIC CHEMISTRY | 2004年 / 69卷 / 23期
关键词：
D O I：
10.1021/jo048837q
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A microwave-assisted synthesis of solid-supported reagents for the acylation of amines has been developed, and the same methodology has been successfully applied to the preparation of acylating agents anchored on different solid supports. Similarly, alcohols, phenols, and thiophenols have been easily acylated using these reagents under microwave irradiation.
引用
收藏
页码：7880 / 7887
页数：8
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