An efficient microwave-assisted Suzuki cross-coupling reaction of imidazo[1,2-a]pyridines in aqueous medium

被引：32
|
作者：
Crozet, Maxime D. [1 ]
Castera-Ducros, Caroline [1 ]
Vanelle, Patrice [1 ]
机构：
[1] Univ Mediterranee, Fac Pharm, CNRS, LCOP,Lab Chim Organ Pharmaceut,UMR 6517, F-13385 Marseille 5, France
来源：
TETRAHEDRON LETTERS | 2006年 / 47卷 / 39期
关键词：
imidazo[1,2-a]pyridines; microwave irradiation; aqueous medium; Suzuki;
D O I：
10.1016/j.tetlet.2006.07.098
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A new simple, rapid and high yielding synthesis of various 6-aryl-2-arylsulfonylmethyl-3-nitroimidazo[1,2-a]pyridines by Suzuki cross-coupling reaction is described using microwave irradiation in aqueous medium without organic co-solvent in the presence of tetrabutylammonium bromide. (c) 2006 Elsevier Ltd. All rights reserved.
引用
收藏
页码：7061 / 7065
页数：5
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