An efficient aqueous microwave-assisted Suzuki-Miyaura cross-coupling reaction in the thiazole series

被引:55
|
作者
Cohen, Anita [1 ]
Crozet, Maxime D.
Rathelot, Pascal
Vanelle, Patrice
机构
[1] Univ Aix Marseille 1, Fac Pharm, Lab Pharmacochim Radicalaire, F-13385 Marseille 05, France
关键词
PALLADIUM-CATALYZED ARYLATION; UNSYMMETRICAL BIARYLS; PROMOTED SYNTHESIS; WATER; ARYL; CHEMISTRY; FUNCTIONALIZATION; TETRAPHENYLBORATE; DERIVATIVES; CYCLIZATION;
D O I
10.1039/b916123f
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
A new simple, rapid and high yielding synthesis of various 5-substituted thiazoles by Suzuki-Miyaura cross-coupling reaction is described using microwave irradiation in aqueous medium without organic co-solvent in the presence of tetrabutylammonium bromide.
引用
收藏
页码:1736 / 1742
页数:7
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