Novel, small molecule inhibitors of HIV-1 integrase

被引:0
|
作者
Wu, J. J. [1 ]
Milot, G. [1 ]
Dandache, S. [1 ]
Gouveia, K. [1 ]
Xiao, Y. [1 ]
Yelle, J. [1 ]
Sevigny, G. [1 ]
Dubois, A. [1 ]
Tian, B. [1 ]
Perron, V. [1 ]
Herbart, D. [1 ]
Stranix, B. R. [1 ]
机构
[1] Ambrilia Biopharma Inc, Montreal, PQ, Canada
关键词
D O I
暂无
中图分类号
R51 [传染病];
学科分类号
100401 ;
摘要
引用
收藏
页码:S8 / S8
页数:1
相关论文
共 50 条
  • [21] Development of a fluorescence-based HIV-1 integrase DNA binding assay for identification of novel HIV-1 integrase inhibitors
    Han, Ying-Shan
    Xiao, Wei-Lie
    Quashie, Peter K.
    Mesplede, Thibault
    Xu, Hongtao
    Deprez, Eric
    Delelis, Olivier
    Pu, Jian-Xin
    Sun, Han-Dong
    Wainberg, Mark A.
    ANTIVIRAL RESEARCH, 2013, 98 (03) : 441 - 448
  • [22] Novel small-molecule compounds which inhibit strand transfer activity of HIV-1 integrase
    Yan, H
    Chiba, T
    Kitamura, Y
    Nishizawa, M
    Fujino, M
    Yamamoto, N
    Sugiura, W
    ANTIVIRAL THERAPY, 2004, 9 (04) : U23 - U23
  • [23] Binding modes of two novel dinucleotide inhibitors of HIV-1 integrase
    Guenther, S
    Nair, V
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2002, 12 (16) : 2233 - 2236
  • [24] Design and synthesis of novel pyrimidone analogues as HIV-1 integrase inhibitors
    Yu, Shenghui
    Sanchez, Tino Wilson
    Liu, Yang
    Yin, Yanzhen
    Neamati, Nouri
    Zhao, Guisen
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (22) : 6134 - 6137
  • [25] Novel HIV-1 integrase inhibitors derived from quinolone antibiotics
    Sato, M
    Motomura, T
    Aramaki, H
    Matsuda, T
    Yamashita, M
    Ito, Y
    Kawakami, H
    Matsuzaki, Y
    Watanabe, W
    Yamataka, K
    Ikeda, S
    Kodama, E
    Matsuoka, M
    Shinkai, H
    JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (05) : 1506 - 1508
  • [26] Novel allosteric inhibitors of HIV-1 integrase on the base of multimodified oligonucleotides
    Zatsepin, T.
    Korolev, S.
    Smolov, M.
    Gottikh, M.
    Agapkina, J.
    FEBS JOURNAL, 2010, 277 : 94 - 94
  • [27] Novel aryl diketo-containing inhibitors of HIV-1 integrase
    Pais, GCG
    Burke, TR
    DRUGS OF THE FUTURE, 2002, 27 (11) : 1101 - 1111
  • [28] Design and synthesis of novel β-diketo derivatives as HIV-1 integrase inhibitors
    Hu, Liming
    Zhang, Sulei
    He, Xianzhuo
    Luo, Zaigang
    Wang, Xiaoli
    Liu, Wei
    Qin, Xuemei
    BIOORGANIC & MEDICINAL CHEMISTRY, 2012, 20 (01) : 177 - 182
  • [29] An Isoquinoline Scaffold as a Novel Class of Allosteric HIV-1 Integrase Inhibitors
    Wilson, Tyler A.
    Koneru, Pratibha C.
    Rebensburg, Stephanie V.
    Lindenberger, Jared J.
    Kobe, Matthew J.
    Cockroft, Nicholas T.
    Adu-Arnpratwum, Daniel
    Larue, Ross C.
    Kvaratskhelia, Mamuka
    Fuchs, James R.
    ACS MEDICINAL CHEMISTRY LETTERS, 2019, 10 (02): : 215 - 220
  • [30] Multimerization selective inhibitors of HIV-1 integrase
    Kvaratskhelia, Mamuka
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250