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- [1] An Isoquinoline Scaffold as a Novel Class of Allosteric HIV-1 Integrase Inhibitors[J]. ACS MEDICINAL CHEMISTRY LETTERS, 2019, 10 (02): : 215 - 220Wilson, Tyler A.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USAKoneru, Pratibha C.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Div Infect Dis, Sch Med, Aurora, CO 80045 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USARebensburg, Stephanie V.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Div Infect Dis, Sch Med, Aurora, CO 80045 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USALindenberger, Jared J.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Div Infect Dis, Sch Med, Aurora, CO 80045 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USAKobe, Matthew J.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Pharmaceut & Pharmaceut Chem, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USACockroft, Nicholas T.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USAAdu-Arnpratwum, Daniel论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USALarue, Ross C.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Pharmaceut & Pharmaceut Chem, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USAKvaratskhelia, Mamuka论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Div Infect Dis, Sch Med, Aurora, CO 80045 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USAFuchs, James R.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA
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- [3] Indole-based allosteric inhibitors of HIV-1 integrase[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 26 (19) : 4748 - 4752Patel, Pratiq A.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Dept Chem, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAKvaratskhelia, Nina论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Pharmaceut & Pharmaceut Chem, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAMansour, Yara论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USA Helwan Univ, Dept Organ Pharmaceut Chem, Fac Pharm, Cairo, Egypt Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAAntwi, Janet论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAFeng, Lei论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Pharmaceut & Pharmaceut Chem, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAKoneru, Pratibha论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Pharmaceut & Pharmaceut Chem, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAKobe, Mathew J.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Pharmaceut & Pharmaceut Chem, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAJena, Nivedita论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAShi, Guqin论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAMohamed, Mosaad S.论文数: 0 引用数: 0 h-index: 0机构: Helwan Univ, Dept Organ Pharmaceut Chem, Fac Pharm, Cairo, Egypt Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USALi, Chenglong论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAKessl, Jacques J.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Pharmaceut & Pharmaceut Chem, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USAFuchs, James R.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Chem & Pharmacognosy, Coll Pharm, Columbus, OH 43210 USA
- [4] Design and synthesis of novel and potent allosteric HIV-1 integrase inhibitors with a spirocyclic moiety[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 110Adachi, Kaoru论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanManabe, Tomoyuki论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Innovat Implementat Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanYamasaki, Takayuki论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Dept Res Planning, Preclin, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanSuma, Akira论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Innovat Implementat Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanOrita, Takuya论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanFuruzono, Tomoko论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanAdachi, Tsuyoshi论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanOhata, Yoshitsugu论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Biol Pharmacol Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanAkiyama, Yoshiyuki论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, DMPK Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanMiyazaki, Susumu论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan
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- [7] Multimode, Cooperative Mechanism of Action of Allosteric HIV-1 Integrase Inhibitors[J]. JOURNAL OF BIOLOGICAL CHEMISTRY, 2012, 287 (20) : 16801 - 16811Kessl, Jacques J.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Comprehens Canc, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USAJena, Nivedita论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USAKoh, Yasuhiro论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Canc Immunol & AIDS, Boston, MA 02215 USA Harvard Univ, Sch Med, Dept Med, Boston, MA 02215 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USATaskent-Sezgin, Humeyra论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Vet Biosci, Ctr Retrovirus Res, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USA论文数: 引用数: h-index:机构:Feng, Lei论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Comprehens Canc, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USAde Silva, Suresh论文数: 0 引用数: 0 h-index: 0机构: NCI, HIV Drug Resistance Program, Frederick, MD 21702 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USAWu, Li论文数: 0 引用数: 0 h-index: 0机构: NCI, HIV Drug Resistance Program, Frederick, MD 21702 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USALe Grice, Stuart F. J.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Vet Biosci, Ctr Retrovirus Res, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USAEngelman, Alan论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Canc Immunol & AIDS, Boston, MA 02215 USA Harvard Univ, Sch Med, Dept Med, Boston, MA 02215 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USAFuchs, James R.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USAKvaratskhelia, Mamuka论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Comprehens Canc, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Ctr Retrovirus Res, Columbus, OH 43210 USA
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