Combinatorial Synthesis of 3,5-Dimethylene Substituted 1,2,4-Triazoles

被引：0
|
作者：
Woodard, Scott S. [1 ]
Jerome, Kevin D. [1 ]
机构：
[1] Pfizer Inc, Global Res & Dev, Med & Parallel Chem, Chesterfield, MO 63017 USA
来源：
COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING | 2011年 / 14卷 / 02期
关键词：
Cyclizations; combinatorial chemistry; 1,2,4-triazoles; Pinner reaction; hydrazides; imidates; 3,5-DISUBSTITUTED 1,2,4-TRIAZOLES; MIT IMIDSAUREESTERN; ANTIBACTERIAL; CYCLIZATION; ANTAGONISTS; AGENTS; ROUTE;
D O I：
暂无
中图分类号：
Q5 [生物化学];
学科分类号：
071010 ; 081704 ;
摘要：
Combinatorial cyclizations of imidates and hydrazides with methylene linked R groups, generated from the corresponding nitriles and carboxylic acids, respectively, provided a large library of 3,5-dimethylene substituted 1,2,4-trizoles. [GRAPHICS] .
引用
收藏
页码：132 / 137
页数：6
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