共 50 条
- [31] Synthetic studies on selective type IV phosphodiesterase(PDE IV) inhibitors. III.[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1998, 216 : U215 - U215Iwata, M论文数: 0 引用数: 0 h-index: 0机构: Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanTakayama, K论文数: 0 引用数: 0 h-index: 0机构: Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanHisamichi, H论文数: 0 引用数: 0 h-index: 0机构: Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanKubota, H论文数: 0 引用数: 0 h-index: 0机构: Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanKawano, N论文数: 0 引用数: 0 h-index: 0机构: Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanAoki, M论文数: 0 引用数: 0 h-index: 0机构: Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanIsomura, Y论文数: 0 引用数: 0 h-index: 0机构: Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Yamanouchi Pharmaceut Co Ltd, Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan
- [32] Nitrogen-bridged substituted 8-arylquinolines as potent PDE IV inhibitors[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (10) : 2608 - 2612Lacombe, P论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaDeschênes, D论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaDubé, D论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaDubé, L论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaGallant, M论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaMacdonald, D论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaMastracchlo, A论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaPerrier, H论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaCharleson, S论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaHuang, Z论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaLaliberté, F论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaLiu, S论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaMancini, JA论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaMasson, P论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaSalem, M论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaStyhler, A论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, CanadaGirard, Y论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada
- [33] Novel, potent and selective angiotensin IV short analogues[J]. JOURNAL OF PEPTIDE SCIENCE, 2008, 14 (08) : 143 - 144Lukaszuk, Aneta论文数: 0 引用数: 0 h-index: 0机构: Vrije Univ Brussels, Brussels, Belgium Vrije Univ Brussels, Brussels, BelgiumDemaegdt, Heidi论文数: 0 引用数: 0 h-index: 0机构: Vrije Univ Brussels, Brussels, Belgium Vrije Univ Brussels, Brussels, BelgiumKaroyan, Philippe论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 06, F-75252 Paris 05, France Vrije Univ Brussels, Brussels, BelgiumVanderheyden, Patrick论文数: 0 引用数: 0 h-index: 0机构: Vrije Univ Brussels, Brussels, Belgium Vrije Univ Brussels, Brussels, BelgiumVauquelin, Georges论文数: 0 引用数: 0 h-index: 0机构: Vrije Univ Brussels, Brussels, Belgium Vrije Univ Brussels, Brussels, BelgiumTourwe, Dirk论文数: 0 引用数: 0 h-index: 0机构: Vrije Univ Brussels, Brussels, Belgium Vrije Univ Brussels, Brussels, Belgium
- [34] First Optimization of Novel, Potent, Selective PDE11A4 Inhibitors for Age-Related Cognitive Decline[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (21) : 14597 - 14608Mahmood, Shams ul论文数: 0 引用数: 0 h-index: 0机构: Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USA Montclair State Univ, Sokol Inst Pharmaceut Life Sci, Montclair, NJ 07043 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USALozano Gonzalez, Mariana论文数: 0 引用数: 0 h-index: 0机构: Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USA Montclair State Univ, Sokol Inst Pharmaceut Life Sci, Montclair, NJ 07043 USA Inst Chem, Coyoacan 04510, DF, Mexico Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USATummalapalli, Sreedhar论文数: 0 引用数: 0 h-index: 0机构: Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USA Montclair State Univ, Sokol Inst Pharmaceut Life Sci, Montclair, NJ 07043 USA A1 Biochem Labs, 5598 Marvin K Moss Lane, Wilmington, NC 28409 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USAEberhard, Jeremy论文数: 0 引用数: 0 h-index: 0机构: Boston Coll, Dept Biol, Chestnut Hill, MA 02467 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USALy, Judy论文数: 0 引用数: 0 h-index: 0机构: Boston Coll, Dept Biol, Chestnut Hill, MA 02467 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USAHoffman, Charles论文数: 0 引用数: 0 h-index: 0机构: Boston Coll, Dept Biol, Chestnut Hill, MA 02467 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USAKelly, Michy论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Med, Dept Anat & Neurobiol, Baltimore, MD 21201 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USAGordon, John论文数: 0 引用数: 0 h-index: 0机构: Temple Univ, Moulder Ctr Drug Discovery Res, Philadelphia, PA 19140 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USAColussi, Dennis论文数: 0 引用数: 0 h-index: 0机构: Temple Univ, Moulder Ctr Drug Discovery Res, Philadelphia, PA 19140 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USAChilders, Wayne论文数: 0 引用数: 0 h-index: 0机构: Temple Univ, Moulder Ctr Drug Discovery Res, Philadelphia, PA 19140 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USARotella, David论文数: 0 引用数: 0 h-index: 0机构: Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USA Montclair State Univ, Sokol Inst Pharmaceut Life Sci, Montclair, NJ 07043 USA Montclair State Univ, Dept Chem & Biochem, Montclair, NJ 07043 USA
- [35] A novel series of potent and selective PDE5 inhibitors with potential for high and dose-independent oral bioavailability[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (12) : 3581 - 3594Allerton, Charlotte M. N.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandBarber, Christopher G.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandBeaumont, Kevin C.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandBrown, David G.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandCole, Susan M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandEllis, David论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandLane, Charlotte A. L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandMaw, Graham N.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandMount, Natalie M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandRawson, David J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandRobinson, Colin M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandStreet, Stephen D. A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, EnglandSummerhill, Nicholas W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Chem, Sandwich CT13 9NJ, Kent, England
- [36] Novel trans-2-aryl-cyclopropylamine analogues as potent and selective dipeptidyl peptidase IV inhibitors[J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2009, 17 (06) : 2388 - 2399Tsai, Ting-Yueh论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanHsu, Tsu论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanChen, Chiung-Tong论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanCheng, Jai-Hong论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanYeh, Teng-Kuang论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanChen, Xin论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanHuang, Chung-Yu论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanChang, Chung-Nien论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanYeh, Kai-Chia论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanHsieh, Su-Huei论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanChien, Chia-Hui论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanChang, Yi-Wei论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanHuang, Chih-Hsiang论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanHuang, Yu-Wen论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanHuang, Chen-Lung论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanWu, Ssu-Hui论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanWang, Min-Hsien论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanLu, Cheng-Tai论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanChao, Yu-Sheng论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, TaiwanJiaang, Weir-Torn论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan Natl Hlth Res Inst, Div Biotechnol & Pharmaceut Res, Zhunan Town 350, Miaoli Country, Taiwan
- [37] Potent and selective azetidine-based dipeptidyl peptidase IV (DPP IV) inhibitors[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 229 : U145 - U146Li, WX论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAOliver, E论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USARojas, C论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USALauter, S论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAThomas, B论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USABelyakov, S论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USA
- [38] Pyrimidinylpyrroloquinolones as highly potent and selective PDE5 inhibitors for treatment of erectile dysfunction[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2002, 45 (19) : 4094 - 4096Sui, ZH论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USAGuan, JH论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USAMacielag, MJ论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USAJiang, WQ论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USAZhang, SY论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USAQiu, YH论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USAKraft, P论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USABhattacharjee, S论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USAJohn, TM论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USAHaynes-Johnson, D论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USAClancy, J论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery, Raritan, NJ 08869 USA
- [39] Discovery of potent, selective, bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model, Part I: Transformation of selective pyrazolodiazepinone phosphodiesterase 4 (PDE4) inhibitors into selective PDE2 inhibitors[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (11) : 3438 - 3442Plummer, Mark S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USACornicelli, Joseph论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Inflammat Pharmacol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USARoark, Howard论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USASkalitzky, Donald J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAStankovic, Charles J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Pharmacodynam & Drug Metab, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USABove, Susan论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Inflammat Pharmacol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAPandit, Jayvardhan论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Technol, Groton, CT 06340 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAGoodman, Annise论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAHicks, James论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAShahripour, Aurash论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USABeidler, David论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Inflammat Pharmacol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USALu, Xiao Kang论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Inflammat Pharmacol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USASanchez, Brian论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Inflammat Pharmacol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAWhitehead, Christopher论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USASarver, Ron论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Technol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USABraden, Timothy论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Inflammat Pharmacol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAGowan, Richard论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Inflammat Pharmacol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAShen, Xi Qiang论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Inflammat Pharmacol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAWelch, Katherine论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Inflammat Pharmacol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAOgden, Adam论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Pharmacodynam & Drug Metab, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USASadagopan, Nalini论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Pharmacodynam & Drug Metab, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USABaum, Heidi论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Pharmacodynam & Drug Metab, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USAMiller, Howard论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Pharmacodynam & Drug Metab, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USABanotai, Craig论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Technol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USASpessard, Cindy论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Technol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USALightle, Sandra论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Discovery Technol, Ann Arbor, MI 48105 USA Pfizer Global Res & Dev, Dept Chem, Ann Arbor, MI 48105 USA
- [40] Heteroatom-bridged substituted 8-arylquinolines as potent PDE IV inhibitors.[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 224 : U64 - U64Lacombe, P论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaDeschênes, D论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaDubé, D论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaDubé, L论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaGallant, M论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaMacdonald, D论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaMastracchio, A论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaPerrier, H论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaCharleson, S论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaHuang, Z论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaLaliberté, F论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaMancini, JA论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaMasson, P论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaStyhler, A论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaNicholson, DW论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, CanadaGirard, Y论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Pointe Claire, PQ H9R 4P8, Canada