Synthesis, reactions and antimicrobial activity of some new 1,3,4-oxadiazoles, 1,2,4-triazoles and 1,3,4-thiadiazines derived from pyrazole.

被引：0
|
作者：
Farghaly, AA [1 ]
Vanelle, P
El-Kashef, HS
机构：
[1] Assiut Univ, Fac Sci, Dept Chem, Assiut 71516, Egypt
[2] Fac Pharm Marseille, UMR CNRS 6517, Lab Chim Organ Pharmaceut, F-13385 Marseille, France
来源：
HETEROCYCLIC COMMUNICATIONS | 2005年 / 11卷 / 3-4期
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D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
New 1,3,4-oxadiazoles, 1,2,4-triazoles and 1,3,4-thiadiazines containing a pyrazolyl moiety 7-14 were prepared using ethyl 5-amino-1-phenyl-1H-pyrazole-3-carboxylate 1 as a starting material. The newly synthesized compounds were screened for their in vitro anti-bacterial and anti-fangal activity.
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页码：255 / 262
页数：8
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