Synthesis of pyrrole- and indole-containing nitropropanoates on the basis of β-heteryl-α-nitroacrylates

被引:13
|
作者
Baichurina, L. V. [1 ]
Baichurin, R. I. [1 ]
Aboskalova, N. I. [1 ]
Berestovitskaya, V. M. [1 ]
机构
[1] Herzen Russian State Pedag Univ, St Petersburg 191186, Russia
关键词
ACID;
D O I
10.1134/S1070363210100221
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Synthetic approach to beta-furyl- and beta-thienyl-alpha-nitroacrylates was modified. It was established that these nitroethenes react with pyrrole, N-methylpyrrole, and substituted indole derivatives in the absence of catalyst to afford products of the alkylation of pyrrole C-2 and indole C-3 reaction sites. A possibility of this reaction to proceed under "dry reaction" condition on a silicagel surface was shown.
引用
收藏
页码:2022 / 2026
页数:5
相关论文
共 50 条
  • [1] Synthesis of pyrrole- and indole-containing nitropropanoates on the basis of β-heteryl-α-nitroacrylates
    L. V. Baichurina
    R. I. Baichurin
    N. I. Aboskalova
    V. M. Berestovitskaya
    Russian Journal of General Chemistry, 2010, 80 : 2022 - 2026
  • [2] Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cells
    Rodriguez, Veronica
    Valente, Sergio
    Rovida, Stefano
    Rotili, Dante
    Stazi, Giulia
    Lucidi, Alessia
    Ciossani, Giuseppe
    Mattevi, Andrea
    Botrugno, Oronza A.
    Dessanti, Paola
    Mercurio, Ciro
    Vianello, Paola
    Minucci, Saverio
    Varasi, Mario
    Mai, Antonello
    MEDCHEMCOMM, 2015, 6 (04) : 665 - 670
  • [3] Synthesis of Indole-containing Hexahydrobenzofuranes
    V. M. Berestovitskaya
    O. S. Vasil'eva
    S. M. Aleksandrova
    Russian Journal of Organic Chemistry, 2001, 37 : 1505 - 1506
  • [4] Synthesis of indole-containing hexahydrobenzofuranes
    Berestovitskaya, VM
    Vasil'eva, OS
    Aleksandrova, SM
    RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, 2001, 37 (10) : 1505 - 1506
  • [5] SYNTHESIS AND INVESTIGATION OF INDOLE-CONTAINING POLYARYLATES
    OVSYANNIKOVA, NN
    SAMSONIYA, SA
    VASNEV, VA
    SUVOROV, NN
    VYSOKOMOLEKULYARNYE SOEDINENIYA SERIYA A, 1984, 26 (01): : 189 - 192
  • [6] Indole-containing derivatives of α-pyrrolidone: Synthesis and structure
    Ostroglyadov, E. S.
    Vasil'eva, O. S.
    Aleksandrova, S. M.
    Pelipko, V. V.
    Berestovitskaya, V. M.
    Tyurenkov, I. N.
    Bagmetova, V. V.
    RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2015, 85 (08) : 1838 - 1844
  • [7] SYNTHESIS OF A NEW CLASS OF INDOLE-CONTAINING MACROCYCLES
    BLACK, DS
    CRAIG, DC
    KUMAR, N
    JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1989, (07) : 425 - 426
  • [8] SYNTHESIS AND STUDY OF INDOLE-CONTAINING POLYARYLATES.
    Ovsyannikova, N.N.
    Samsoniya, Sh.A.
    Vasnev, V.A.
    Suvorov, N.N.
    Polymer science USSR, 1984, 26 (01): : 210 - 215
  • [9] Indole-containing derivatives of α-pyrrolidone: Synthesis and structure
    E. S. Ostroglyadov
    O. S. Vasil’eva
    S. M. Aleksandrova
    V. V. Pelipko
    V. M. Berestovitskaya
    I. N. Tyurenkov
    V. V. Bagmetova
    Russian Journal of General Chemistry, 2015, 85 : 1838 - 1844
  • [10] Catalytic asymmetric synthesis of indole-containing macrocycles
    Woods, Philip
    Waring, Michael
    Moss, Thomas
    Dixon, Darren
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250