Synthesis of pyrrole- and indole-containing nitropropanoates on the basis of β-heteryl-α-nitroacrylates

被引：13

作者：

Baichurina, L. V. ^{[1
]}

Baichurin, R. I. ^{[1
]}

Aboskalova, N. I. ^{[1
]}

Berestovitskaya, V. M. ^{[1
]}

机构：

[1] Herzen Russian State Pedag Univ, St Petersburg 191186, Russia

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2010年 / 80卷 / 10期

关键词：

ACID;

D O I：

10.1134/S1070363210100221

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Synthetic approach to beta-furyl- and beta-thienyl-alpha-nitroacrylates was modified. It was established that these nitroethenes react with pyrrole, N-methylpyrrole, and substituted indole derivatives in the absence of catalyst to afford products of the alkylation of pyrrole C-2 and indole C-3 reaction sites. A possibility of this reaction to proceed under "dry reaction" condition on a silicagel surface was shown.

引用

页码：2022 / 2026

页数：5

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