Dissecting physiological roles of estrogen receptor alpha and beta with selective Ligands from protein structure-based design.

被引：0
|
作者：
Hillisch, A
Peters, O
Müller, G
Kosemund, D
Elger, W
Hegele-Hartung, C
Fritzemeier, KH
机构：
[1] EnTec GmbH, Jena, Germany
[2] Jenapharm, Jena, Germany
[3] Schering AG, D-1000 Berlin, Germany
来源：
CANCER EPIDEMIOLOGY BIOMARKERS & PREVENTION | 2005年 / 14卷 / 11期
关键词：
D O I：
暂无
中图分类号：
R73 [肿瘤学];
学科分类号：
100214 ;
摘要：
引用
收藏
页码：2780S / 2781S
页数：2
相关论文
共 50 条
  • [1] Dissecting physiological roles of estrogen receptor α and β with potent selective ligands from structure-based design
    Hillisch, A
    Peters, O
    Kosemund, D
    Müller, G
    Walter, A
    Schneider, B
    Reddersen, G
    Elger, W
    Fritzemeier, KH
    [J]. MOLECULAR ENDOCRINOLOGY, 2004, 18 (07) : 1599 - 1609
  • [2] Structure-based design of estrogen receptor-β selective ligands
    Manas, ES
    Unwalla, RJ
    Xu, ZB
    Malamas, MS
    Miller, CP
    Harris, HA
    Hsiao, C
    Akopian, T
    Hum, WT
    Malakian, K
    Wolfrom, S
    Bapat, A
    Bhat, RA
    Stahl, ML
    Somers, WS
    Alvarez, JC
    [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2004, 126 (46) : 15106 - 15119
  • [3] Structure-based design of estrogen receptor-beta selective compounds
    Malamas, Michael S.
    Harris, Heather A.
    Keith, Jim
    McDevitt, Bob
    Gunawan, Iwan
    Manas, Eric
    Miller, Christopher P.
    Mewshaw, Richard E.
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 232 : 310 - 310
  • [4] Structure-based design of selective nuclear hormone receptor ligands
    Magolda, RL
    Fensome, A
    Harnish, D
    Harris, HA
    Keith, JC
    Malamas, MS
    Manas, E
    Mewshaw, RE
    Olland, A
    Somers, WS
    Steffan, RJ
    Trybulski, EJ
    Unwalla, RJ
    Winneker, RC
    Wrobel, L
    Xu, ZB
    Zhang, PW
    Zhang, Z
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 230 : U2639 - U2640
  • [5] Design and synthesis of selective estrogen modulators and estrogen receptor beta selective ligands.
    Collini, M
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2003, 226 : U220 - U221
  • [6] Protein structure-based design, synthesis strategy and in vitro pharmacological characterization of estrogen receptor α and β selective compounds
    Hillisch, A
    Peters, O
    Kosemund, D
    Müller, G
    Walter, A
    Elger, W
    Fritzemeier, KH
    [J]. NEW MOLECULAR MECHANISMS OF ESTROGEN ACTION AND THEIR IMPACT ON FUTURE PERSPECTIVES IN ESTROGEN THERAPY, 2004, 46 : 47 - 62
  • [7] Structure-based design of adenosine receptor ligands
    Jacobson, Kenneth A.
    Stevens, Raymond C.
    Abagyan, Ruben
    Deflorian, Francesca
    Gao, Zhan-Guo
    Gakh, Andrei A.
    Tosh, Dilip K.
    Kumar, T. S.
    Xu, Fei
    Katritch, Vsevolod
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 243
  • [8] Selective ligands of estrogen receptor β discovered using pharmacophore mapping and structure-based virtual screening
    Chen, Lei
    Wu, Dang
    Bian, Han-ping
    Kuang, Guang-lin
    Jiang, Jing
    Li, Wei-hua
    Liu, Gui-xia
    Zou, Shi-en
    Huang, Jin
    Tang, Yun
    [J]. ACTA PHARMACOLOGICA SINICA, 2014, 35 (10) : 1333 - 1341
  • [9] Selective ligands of estrogen receptor β discovered using pharmacophore mapping and structure-based virtual screening
    Lei Chen
    Dang Wu
    Han-ping Bian
    Guang-lin Kuang
    Jing Jiang
    Wei-hua Li
    Gui-xia Liu
    Shi-en Zou
    Jin Huang
    Yun Tang
    [J]. Acta Pharmacologica Sinica, 2014, 35 : 1333 - 1341
  • [10] Structure-based design of bitopic ligands for the µ-opioid receptor
    Abdelfattah Faouzi
    Haoqing Wang
    Saheem A. Zaidi
    Jeffrey F. DiBerto
    Tao Che
    Qianhui Qu
    Michael J. Robertson
    Manish K. Madasu
    Amal El Daibani
    Balazs R. Varga
    Tiffany Zhang
    Claudia Ruiz
    Shan Liu
    Jin Xu
    Kevin Appourchaux
    Samuel T. Slocum
    Shainnel O. Eans
    Michael D. Cameron
    Ream Al-Hasani
    Ying Xian Pan
    Bryan L. Roth
    Jay P. McLaughlin
    Georgios Skiniotis
    Vsevolod Katritch
    Brian K. Kobilka
    Susruta Majumdar
    [J]. Nature, 2023, 613 : 767 - 774
12345