Structure-based design of selective nuclear hormone receptor ligands

被引：0
|
作者：
Magolda, RL
Fensome, A
Harnish, D
Harris, HA
Keith, JC
Malamas, MS
Manas, E
Mewshaw, RE
Olland, A
Somers, WS
Steffan, RJ
Trybulski, EJ
Unwalla, RJ
Winneker, RC
Wrobel, L
Xu, ZB
Zhang, PW
Zhang, Z
机构：
[1] Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USA
[2] Wyeth Res, Cardiovasc Metab Dis, Princeton, NJ 08543 USA
[3] Wyeth Res, Womens Hlth Res Inst, Princeton, NJ 08543 USA
[4] Wyeth Res, Womens Hlth & Musculoskeletal Biol, Princeton, NJ 08543 USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2005年 / 230卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
236-MEDI
引用
收藏
页码：U2639 / U2640
页数：2
相关论文
共 50 条
  • [1] Structure-based design of estrogen receptor-β selective ligands
    Manas, ES
    Unwalla, RJ
    Xu, ZB
    Malamas, MS
    Miller, CP
    Harris, HA
    Hsiao, C
    Akopian, T
    Hum, WT
    Malakian, K
    Wolfrom, S
    Bapat, A
    Bhat, RA
    Stahl, ML
    Somers, WS
    Alvarez, JC
    [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2004, 126 (46) : 15106 - 15119
  • [2] Structure-based design of adenosine receptor ligands
    Jacobson, Kenneth A.
    Stevens, Raymond C.
    Abagyan, Ruben
    Deflorian, Francesca
    Gao, Zhan-Guo
    Gakh, Andrei A.
    Tosh, Dilip K.
    Kumar, T. S.
    Xu, Fei
    Katritch, Vsevolod
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 243
  • [3] Structure-based design of bitopic ligands for the µ-opioid receptor
    Abdelfattah Faouzi
    Haoqing Wang
    Saheem A. Zaidi
    Jeffrey F. DiBerto
    Tao Che
    Qianhui Qu
    Michael J. Robertson
    Manish K. Madasu
    Amal El Daibani
    Balazs R. Varga
    Tiffany Zhang
    Claudia Ruiz
    Shan Liu
    Jin Xu
    Kevin Appourchaux
    Samuel T. Slocum
    Shainnel O. Eans
    Michael D. Cameron
    Ream Al-Hasani
    Ying Xian Pan
    Bryan L. Roth
    Jay P. McLaughlin
    Georgios Skiniotis
    Vsevolod Katritch
    Brian K. Kobilka
    Susruta Majumdar
    [J]. Nature, 2023, 613 : 767 - 774
  • [4] Structure-based drug design for nuclear hormone receptors
    Krystek, SR
    Hamann, LG
    Salvati, ME
    Balog, A
    Hunt, J
    Li, J
    Manfredi, M
    Martinez, R
    Nayeem, A
    Nirsch, A
    Pickering, D
    Schnur, D
    Shan, WF
    Sun, CQ
    Wei, D
    Zhu, H
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 230 : U1294 - U1294
  • [5] Structure-Based Rational Design of Adenosine Receptor Ligands
    Gutierrez-de-Teran, Hugo
    Sallander, Jessica
    Sotelo, Eddy
    [J]. CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2017, 17 (01) : 40 - 58
  • [6] Structure-based design of bitopic ligands for the μ-opioid receptor
    Faouzi, Abdelfattah
    Wang, Haoqing
    Zaidi, Saheem A.
    DiBerto, Jeffrey F.
    Che, Tao
    Qu, Qianhui
    Robertson, Michael J.
    Madasu, Manish K.
    El Daibani, Amal
    Varga, Balazs R.
    Zhang, Tiffany
    Ruiz, Claudia
    Liu, Shan
    Xu, Jin
    Appourchaux, Kevin
    Slocum, Samuel T.
    Eans, Shainnel O.
    Cameron, Michael D.
    Al-Hasani, Ream
    Pan, Ying Xian
    Roth, Bryan L.
    McLaughlin, Jay P.
    Skiniotis, Georgios
    Katritch, Vsevolod
    Kobilka, Brian K.
    Majumdar, Susruta
    [J]. NATURE, 2023, 613 (7945) : 767 - +
  • [7] Dissecting physiological roles of estrogen receptor α and β with potent selective ligands from structure-based design
    Hillisch, A
    Peters, O
    Kosemund, D
    Müller, G
    Walter, A
    Schneider, B
    Reddersen, G
    Elger, W
    Fritzemeier, KH
    [J]. MOLECULAR ENDOCRINOLOGY, 2004, 18 (07) : 1599 - 1609
  • [8] Structure-Based Evolution of Subtype-Selective Neurotensin Receptor Ligands
    Schaab, Carolin
    Kling, Ralf Christian
    Einsiedel, Juergen
    Huebner, Harald
    Clark, Tim
    Seebach, Dieter
    Gmeiner, Peter
    [J]. CHEMISTRYOPEN, 2014, 3 (05): : 206 - 218
  • [9] Structure-Based Design of Potent and Selective Ligands at the Four Adenosine Receptors
    Jespers, Willem
    Oliveira, Ana
    Prieto-Diaz, Ruben
    Majellaro, Maria
    Aqvist, Johan
    Sotelo, Eddy
    Gutierrez-de-Teran, Hugo
    [J]. MOLECULES, 2017, 22 (11):
  • [10] Synergistic approach of structure-based and ligand-based drug design for the development of selective cannabinod receptor ligands
    Robert Günther
    Peter Brust
    [J]. Journal of Cheminformatics, 4 (Suppl 1)
12345