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- [21] Discovery of Potent, Selective, and Orally Bioavailable Small-Molecule Inhibitors of CDK8 for the Treatment of CancerJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (08) : 5439 - 5452Li, Yangguang论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaLiu, Yingtao论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaWu, Jianping论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaLiu, Xiaosong论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaWang, Lin论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaWang, Ju论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaYu, Jiaojiao论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaQi, Hongyun论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaQin, Luoheng论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaDing, Xiao论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaRen, Feng论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaZhavoronkov, Alex论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China
- [22] Discovery of potent and orally available malonyl- CoA decarboxylase inhibitors as cardioprotective agentsJOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (14) : 4055 - 4058Cheng, Jie-Fei论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USAHuang, Yujin论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USAPenuliar, Richard论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USANishimoto, Masahiro论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USALiu, Larry论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USAArrhenius, Thomas论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USAYang, Guang论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USAO'Leary, Eoin论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USABarbosa, Miguel论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USABarr, Rick论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USADyck, Jason R. B.论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USALopaschuk, Gary D.论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USANadzan, Alex M.论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharma USA, LLC, Dept Chem, San Diego, CA 92121 USA
- [23] Design and Discovery of MRTX0902, a Potent, Selective, Brain- Penetrant, and Orally Bioavailable Inhibitor of the SOS1:KRAS Protein-Protein InteractionJOURNAL OF MEDICINAL CHEMISTRY, 2022, : 9678 - 9690Ketcham, John M.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAHaling, Jacob论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAKhare, Shilpi论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USABowcut, Vickie论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USABriere, David M.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USABurns, Aaron C.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAGunn, Robin J.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAIvetac, Anthony论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAKuehler, Jon论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAKulyk, Svitlana论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USALaguer, Jade论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USALawson, J. David论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAMoya, Krystal论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USANguyen, Natalie论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USARahbaek, Lisa论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USASaechao, Barbara论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USASmith, Christopher R.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USASudhakar, Niranjan论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAThomas, Nicole C.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAVegar, Laura论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAVanderpool, Darin论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAWang, Xiaolun论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAYan, Larry论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAOlson, Peter论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAChristensen, James G.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USAMarx, Matthew A.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA 92121 USA Mirati Therapeut, San Diego, CA 92121 USA
- [24] Discovery of RGT-018: A potent, selective and orally bioavailable SOS1 inhibitor for mutant KRAS-driven cancersCANCER RESEARCH, 2023, 83 (07)Xiao, Fei论文数: 0 引用数: 0 h-index: 0Wang, Kailiang论文数: 0 引用数: 0 h-index: 0Wang, Xinjuan论文数: 0 引用数: 0 h-index: 0Li, Huijuan论文数: 0 引用数: 0 h-index: 0Hu, Zhilong论文数: 0 引用数: 0 h-index: 0Huang, Wei论文数: 0 引用数: 0 h-index: 0Ren, Xiaoming论文数: 0 引用数: 0 h-index: 0Feng, Teng论文数: 0 引用数: 0 h-index: 0Yao, Lili论文数: 0 引用数: 0 h-index: 0Lin, Jing论文数: 0 引用数: 0 h-index: 0Li, Chunlai论文数: 0 引用数: 0 h-index: 0Mei, Liufeng论文数: 0 引用数: 0 h-index: 0Zhang, Zhuanzhuan论文数: 0 引用数: 0 h-index: 0Liu, Yangyang论文数: 0 引用数: 0 h-index: 0Chen, Xi论文数: 0 引用数: 0 h-index: 0Zhu, Xiaotian论文数: 0 引用数: 0 h-index: 0Zhong, Wenge论文数: 0 引用数: 0 h-index: 0Xie, Zhi论文数: 0 引用数: 0 h-index: 0
- [25] Discovery of Potent Small-Molecule Inhibitors of MLL MethyltransferaseACS MEDICINAL CHEMISTRY LETTERS, 2020, 11 (06): : 1348 - 1352Chern, Ting-Rong论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USALiu, Liu论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USAPetrunak, Elyse论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Life Sci Inst, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USAStuckey, Jeanne A.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Life Sci Inst, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Mi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USA论文数: 引用数: h-index:机构:Zhou, Haibin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USALee, Shirley论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USADou, Yali论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Dept Internal Med, Ann Arbor, MI 48109 USA
- [26] Discovery of potent small-molecule inhibitors of lipoprotein(a) formationNATURE, 2024, 629 (8013) : 945 - 950Diaz, Nuria论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Alcobendas, Spain Lilly Res Labs, Alcobendas, SpainPerez, Carlos论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Alcobendas, Spain Lilly Res Labs, Alcobendas, SpainEscribano, Ana Maria论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Alcobendas, Spain Lilly Res Labs, Alcobendas, SpainSanz, Gema论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Alcobendas, Spain Lilly Res Labs, Alcobendas, SpainPriego, Julian论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Alcobendas, Spain Lilly Res Labs, Alcobendas, SpainLafuente, Celia论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Alcobendas, Spain Lilly Res Labs, Alcobendas, SpainBarberis, Mario论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Alcobendas, Spain Lilly Res Labs, Alcobendas, SpainCalle, Luis论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Alcobendas, Spain Lilly Res Labs, Alcobendas, SpainEspinosa, Juan Felix论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Alcobendas, Spain Lilly Res Labs, Alcobendas, SpainPriest, Birgit T.论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Indianapolis, IN 46225 USA Lilly Res Labs, Alcobendas, SpainZhang, Hong Y.论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Indianapolis, IN 46225 USA Lilly Res Labs, Alcobendas, SpainNosie, Amanda K.论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Indianapolis, IN 46225 USA Lilly Res Labs, Alcobendas, SpainHaas, Joseph V.论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Indianapolis, IN 46225 USA Lilly Res Labs, Alcobendas, SpainCannady, Ellen论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Indianapolis, IN 46225 USA Lilly Res Labs, Alcobendas, SpainBorel, Anthony论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Indianapolis, IN 46225 USA Lilly Res Labs, Alcobendas, SpainSchultze, Albert E.论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Indianapolis, IN 46225 USA Lilly Res Labs, Alcobendas, SpainSauder, J. Michael论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, San Diego, CA USA Lilly Res Labs, Alcobendas, SpainHendle, Joerg论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, San Diego, CA USA Lilly Res Labs, Alcobendas, SpainWeichert, Ken论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, San Diego, CA USA Lilly Res Labs, Alcobendas, SpainNicholls, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Victorian Heart Inst, Clayton, Vic, Australia Lilly Res Labs, Alcobendas, SpainMichael, Laura F.论文数: 0 引用数: 0 h-index: 0机构: Lilly Res Labs, Indianapolis, IN 46225 USA Lilly Res Labs, Alcobendas, Spain
- [27] Discovery of orally available and potent MPS1(TTK) kinase inhibitors for anti-cancer drugsCANCER RESEARCH, 2019, 79 (13)Lee, Younho论文数: 0 引用数: 0 h-index: 0机构: NDBio Therapeut, Incheon, South Korea NDBio Therapeut, Incheon, South KoreaKang, Juhee论文数: 0 引用数: 0 h-index: 0机构: NDBio Therapeut, Incheon, South Korea NDBio Therapeut, Incheon, South KoreaKang, Sein论文数: 0 引用数: 0 h-index: 0机构: NDBio Therapeut, Incheon, South Korea NDBio Therapeut, Incheon, South KoreaKim, Hyunkyung论文数: 0 引用数: 0 h-index: 0机构: NDBio Therapeut, Incheon, South Korea NDBio Therapeut, Incheon, South KoreaSeo, Kyung-ah论文数: 0 引用数: 0 h-index: 0机构: NDBio Therapeut, Incheon, South Korea NDBio Therapeut, Incheon, South KoreaChoi, Jieun论文数: 0 引用数: 0 h-index: 0机构: Voronoi, Incheon, South Korea NDBio Therapeut, Incheon, South KoreaAhn, Jaeyoung论文数: 0 引用数: 0 h-index: 0机构: Voronoi, Incheon, South Korea NDBio Therapeut, Incheon, South KoreaSon, Jung Beom论文数: 0 引用数: 0 h-index: 0机构: NDBio Therapeut, Incheon, South Korea NDBio Therapeut, Incheon, South KoreaKim, Nam Doo论文数: 0 引用数: 0 h-index: 0机构: NDBio Therapeut, Incheon, South Korea NDBio Therapeut, Incheon, South Korea
- [28] Discovery of potent small molecule inhibitors of Wnt-dependent transcriptionABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248Mallinger, Aurelie论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandCrumpler, Simon论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandPichowicz, Mark论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandWaalboer, Dennis论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandRaynaud, Florence论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandRohdich, Felix论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandGeorgi, Katrin论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandStubbs, Mark论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandAherne, Wynne论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandDale, Trevor论文数: 0 引用数: 0 h-index: 0机构: Cardiff Univ, Sch Biosci, Cardiff CF10 3AX, S Glam, Wales Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandWienke, Dirk论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandStieber, Frank论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandSchiemann, Kai论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, EnglandBlagg, Julian论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW3 6JB, England
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