REDUCTIVE N-MONOALKYLATION OF PRIMARY AROMATIC-AMINES

被引：1
|
作者：
VERARDO, G [1 ]
GIUMANINI, AG [1 ]
STRAZZOLINI, P [1 ]
POIANA, M [1 ]
机构：
[1] UNIV UDINE,DEPT CHEM SCI & TECHNOL,I-33100 UDINE,ITALY
来源：
SYNTHESIS-STUTTGART | 1993年 / 01期
关键词：
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Primary aromatic amines 1 with a variety of ring substituents are easily converted to their N-monoalkyl derivatives 3 by a simple variation of the sodium borohydride/sulfuric acid/carbonyl compound procedure previously described for their N-permethylations. The procedure is suitable for the alpha-monodeuterium labelling of the new N-substituent.
引用
下载
收藏
页码：121 / 125
页数：5
相关论文
共 50 条
  • [41] REACTION OF ARYLDICHLOROPHOSPHINES AND ARYL DICHLOROPHOSPHITES WITH PRIMARY AROMATIC-AMINES
    TRISHIN, YG
    CHISTOKLETOV, VN
    PETROV, AA
    ZHURNAL OBSHCHEI KHIMII, 1979, 49 (01): : 48 - 53
  • [42] PRIMARY SENSITIVITY TO SULFONAMIDE AND SECONDARY SENSITIZATION TO AROMATIC-AMINES
    RUDZKI, E
    REBANDEL, P
    CONTACT DERMATITIS, 1987, 17 (01) : 49 - 49
  • [43] NEW INTERNAL INDICATORS FOR DETERMINING PRIMARY AROMATIC-AMINES
    ELSEBAI, AI
    BELTAGY, YA
    SOLIMAN, R
    PHARMAZIE, 1971, 26 (10): : 615 - &
  • [44] SPECTROPHOTOMETRIC DETERMINATION OF PRIMARY AROMATIC-AMINES USING SYRINGALDEHYDE
    SASTRY, CSP
    RAO, BG
    SASTRY, BS
    JOURNAL OF THE INDIAN CHEMICAL SOCIETY, 1986, 63 (11) : 1006 - 1007
  • [45] THE OXIDATION OF PRIMARY AROMATIC-AMINES WITH POTASSIUM FERRICYANIDE AND KOH
    LEYVA, E
    CRUZ, E
    VALLE, LE
    MONREAL, E
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1994, 208 : 346 - ORGN
  • [46] MOLECULAR COMPLEXES OF CUMENYL HYDROPEROXIDE WITH PRIMARY AROMATIC-AMINES
    ALEKSANDROV, YA
    VYSHINSKII, NN
    SOLOVEVA, EI
    MOROZOV, OS
    SULDIN, BV
    ZHURNAL OBSHCHEI KHIMII, 1975, 45 (03): : 681 - 684
  • [47] NEW SPECTROPHOTOMETRIC METHOD FOR THE DETERMINATION OF PRIMARY AROMATIC-AMINES
    KRISHNA, RR
    SASTRY, CSP
    TALANTA, 1979, 26 (09) : 861 - 865
  • [48] ALKYLTHIO AROMATIC-AMINES
    RANKEN, PF
    MCKINNIE, BG
    JOURNAL OF ORGANIC CHEMISTRY, 1989, 54 (12): : 2985 - 2988
  • [49] HETEROCYCLOALKYLATION OF AROMATIC-AMINES
    IVANOV, GE
    PAVLYUK, GV
    UKRAINSKII KHIMICHESKII ZHURNAL, 1988, 54 (08): : 872 - 876
  • [50] RADICAL PHTHALIMIDATION OF AROMATIC-COMPOUNDS BY PHOTOLYSIS OF N-TOSYLOXYPHTHALIMIDE - ROUTE TO PRIMARY AROMATIC-AMINES
    CADOGAN, JIG
    ROWLEY, AG
    JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1975, (11): : 1069 - 1071
12345