REDUCTIVE N-MONOALKYLATION OF PRIMARY AROMATIC-AMINES

被引：1

作者：

VERARDO, G ^{[1
]}

GIUMANINI, AG ^{[1
]}

STRAZZOLINI, P ^{[1
]}

POIANA, M ^{[1
]}

机构：

[1] UNIV UDINE,DEPT CHEM SCI & TECHNOL,I-33100 UDINE,ITALY

来源：

SYNTHESIS-STUTTGART | 1993年 / 01期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Primary aromatic amines 1 with a variety of ring substituents are easily converted to their N-monoalkyl derivatives 3 by a simple variation of the sodium borohydride/sulfuric acid/carbonyl compound procedure previously described for their N-permethylations. The procedure is suitable for the alpha-monodeuterium labelling of the new N-substituent.

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页码：121 / 125

页数：5

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