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REDUCTIVE N-MONOALKYLATION OF PRIMARY AROMATIC-AMINES

被引：1
|
作者：
VERARDO, G [1 ]
GIUMANINI, AG [1 ]
STRAZZOLINI, P [1 ]
POIANA, M [1 ]
机构：
[1] UNIV UDINE,DEPT CHEM SCI & TECHNOL,I-33100 UDINE,ITALY
来源：
SYNTHESIS-STUTTGART | 1993年 / 01期
关键词：
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Primary aromatic amines 1 with a variety of ring substituents are easily converted to their N-monoalkyl derivatives 3 by a simple variation of the sodium borohydride/sulfuric acid/carbonyl compound procedure previously described for their N-permethylations. The procedure is suitable for the alpha-monodeuterium labelling of the new N-substituent.
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页码：121 / 125
页数：5
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