SYNTHESIS AND ANTIBACTERIAL ACTIVITY OF SOME NEW PYRIDYL DIARYLSULFIDE AND DIARYLSULFONES

被引：6

作者：

ELEZBAWY, SR ^{[1
]}

ALSHAIKH, MA ^{[1
]}

机构：

[1] GIRLS COLL,DEPT CHEM,JEDDAH,SAUDI ARABIA

来源：

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 1990年 / 48卷 / 1-4期

关键词：

4-thiazolidinones; antibacterial activity diarylsulfide and diaryIsulfone; pyridines; Synthesis;

D O I：

10.1080/10426509008045887

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Condensation of isonicotinaldehyde with 4-aminodiphenyl sulfides I and/or sulfones II gave 4-[N-[p-(diaryl/thio)]formimidoyl]-pyridine III and/or 4-[N-[p-(diarylsulfonyl)]-formimidoyl]pyridine IV. Cyclocondensation of mercaptoacetic acid on III and IV gave 3-[p-(diarylthio)]-2-(4-pyridyl)-4-thiazolidinones V and 3-[p-(diarylsulfonyl)]-2-(4-pyridyl)-4-thiazolidinones VI respectively. (Hetero/arylthio)-N-(6-methyl-2-pyridyl)-acetamides VIII have been synthesised via interaction of 6-methyi-2-chloroacetamido-pyridine VII with heterocyclic and/or aromatic mercaptans. Reaction of VII with piperidine and/or morpholine affords (IX). Biological activities of these compounds were tested. © 1990, Taylor & Francis Group. All rights reserved.

引用

页码：111 / 116

页数：6

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