ELECTROCHEMICAL AND ANTIBACTERIAL BEHAVIOR OF DERIVATIVES OF (1S, 2S) - 2 AMINO- 1- (4-NITROPHENYL) - PROPANE-1,3-DIOL

被引:0
|
作者
Cristea, Cecilia [1 ]
Voiculescu, G. [2 ]
Jitaru, Maria [2 ]
Moinet, C. [3 ]
机构
[1] Univ Med & Pharm Iuliu Hatieganu, Fac Pharm, Dept Chim Analyt, 4 Rue Pasteur, Cluj Napoca 400349, Romania
[2] Univ Babes Bolyai Cluj Napoca, Lab Assoc Francophone, Cluj Napoca 400028, Romania
[3] Univ Rennes 1, Inst Chim, Lab Electrochim & Organometall, F-35042 Rennes, France
关键词
electrosynthesis; hydroxylamines; nitrosoderivatives; redox cell;
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Derivatives of (1S, 2S)-2-amino-1-(4-nitrophenyl)propane-1,3-diol were studied because of their potential biological activity. Using the electrogenerated intermediates (hydroxylamine and nitroso derivatives) N-sulphonylphenylhydroxylamines and benzoxazine diones were obtained with good yields. Their antibacterial activity was investigated on several gram-negative and gram-positive bacilli by two techniques: broth-dilution method and agar-dilution method.
引用
收藏
页码:209 / 216
页数:8
相关论文
共 50 条
  • [21] (1S,2S)-1-(2-bromo-4-hydroxy-3,5-dimethoxyphenyl)propane-1,2,3-triol
    Chand, Satish
    Willis, Anthony C.
    ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2007, 63 : O4866 - U6535
  • [22] 2-{(E)-1-[2-(4-Nitrophenyl) hydrazin-1-ylidene] ethyl}benzene-1,3-diol
    Howie, R. Alan
    Wardell, James L.
    Wardell, Solange M. S. V.
    Tiekink, Edward R. T.
    ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2012, 68 : O685 - U1962
  • [23] STRUCTURE OF 1-(4-NITROPHENYL)PYRROLE, 1-(4-NITROPHENYL)IMIDAZOLE, 1-(4-NITROPHENYL)PYRAZOLE AND 1-(4-NITROPHENYL)1,2,4-TRIAZOLE DERIVATIVES
    ISHIHARA, M
    TONOGAKI, M
    OHBA, S
    SAITO, Y
    OKAZAKI, M
    KATOH, T
    KAMIYAMA, K
    ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS, 1992, 48 : 184 - 188
  • [24] A highly efficient chemoselective cyclocondensation of threo-(1S,2S)-2-amino-1-(4-nitrophenyl)-1,3-propaiiediol with ketones and isomerization of the condensates
    Shan, ZX
    Wan, BY
    Wang, GP
    HELVETICA CHIMICA ACTA, 2002, 85 (04) : 1062 - 1068
  • [25] Synthesis of isomeric 2-oxazolidinones from (1R,2R)-and (1S,2S)-2-amino-1-(4-nitrophenyl)-1,3-propanediols
    Madesclaire M.
    Zaitsev V.P.
    Zaitseva J.V.
    Sharipova S.Kh.
    Chemistry of Heterocyclic Compounds, 2007, 43 (10) : 1325 - 1332
  • [26] Synthesis of isomeric 2-oxazolidinones from (1R,2R)- and (1S,2S)-2-amino-1-(4-nitrophenyl)-1,3-propanediols
    Madesclaire, M.
    Zaitsev, V. P.
    Zaitseva, J. V.
    Sharipova, S. Kh.
    KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII, 2007, (10): : 1562 - 1570
  • [27] threo-2-(2,6-Dimethoxyphenoxy)-1-(4-ethoxy-3-methoxyphenyl)propane-1,3-diol
    Ishizuka, Kentaro
    Ando, Daisuke
    Watanabe, Takashi
    Nakamura, Masaharu
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2009, 65 : O1389 - U2860
  • [28] Synthesis and Anti-MAO Activity of Alkylation Products of 2-Aminobenzamide, 2-Amino-1-(4-nitrophenyl)propane-1,3-diol, and Some Amino Acids with Mono- and Bis-β-aminoketones
    N. Z. Akopyan
    A. G. Agababyan
    Z. A. Ovasyan
    A. U. Isakhanyan
    A. S. Grigoryan
    K. G. Navoyan
    G. V. Gasparyan
    H. A. Panosyan
    Russian Journal of General Chemistry, 2022, 92 : 925 - 931
  • [29] Synthesis and Anti-MAO Activity of Alkylation Products of 2-Aminobenzamide, 2-Amino-1-(4-nitrophenyl)propane-1,3-diol, and Some Amino Acids with Mono- and Bis-β-aminoketones
    Akopyan, N. Z.
    Agababyan, A. G.
    Ovasyan, Z. A.
    Isakhanyan, A. U.
    Grigoryan, A. S.
    Navoyan, K. G.
    Gasparyan, G., V
    Panosyan, H. A.
    RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2022, 92 (06) : 925 - 931
  • [30] Regioselectivity of interaction between paraformaldehyde and (1S,2S)-2-aryl(hetaryl) methylamino-1-(4-nitrophenyl)-1,3-propanediols
    Kukle, Z
    Madeskler, M
    Leal, F
    Zaitsev, VP
    Sharipova, SK
    KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII, 1999, (04): : 536 - 541