Synthesis and pharmacological activity of N-[β-(para-substituted benzoyl)ethyl]isoleucine and -methionine

被引：0

作者：

Agababyan A.G. ^{[1
]}

Isakhanyan A.Y. ^{[1
]}

Papoyan O.A. ^{[1
]}

Tumadzhyan A.E. ^{[1
]}

Balasanyan A.S. ^{[1
]}

Gevorgyan G.A. ^{[1
]}

机构：

[1] Mndzhoyan Institute of Fine Organic Chemistry, National Academy of Sciences of Armenia, Yerevan

来源：

Pharmaceutical Chemistry Journal | 2005年 / 39卷 / 7期

关键词：

Ethyl; Organic Chemistry; Hydrochloride; Methionine; Antiinflammatory Activity;

D O I：

10.1007/s11094-005-0156-2

中图分类号：

学科分类号：

摘要：

A series of N-[β-(p-substituted benzoyl)ethyl]-isoleucine and -methionine derivatives have been synthesized via the alkylation of amino acids with p-substituted β-diethylaminopropiophenone hydrochlorides. Some of the synthesized compounds possess significant antiinflammatory activity. © 2005 Springer Science+Business Media, Inc.

引用

页码：364 / 366

页数：2

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