First cascade Mitsunobu reactions for the synthesis of 2-benzoxazole-N-phenyl and 2-benzimidazole-N-phenyl derivatives

被引：0
|
作者：
Yu Yan
Qifei Zhong
Nan Zhao
Gang Liu
机构：
[1] Institute of Materia Medica,Tsinghua
[2] Chinese Academy of Medical Sciences and Peking Union Medical College,Peking Center for Life Sciences and Department of Pharmacology and Pharmaceutical Sciences, School of Medicine
[3] Tsinghua University,undefined
来源：
Molecular Diversity | 2012年 / 16卷
关键词：
Cascade Mitsunobu reactions; Benzoxazole; Benzimidazole;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
An efficient method has been developed via cascade Mitsunobu reactions to synthesize 2-benzoxazole-N-phenyl and 2-benzimidazole-N-phenyl derivatives, which are common structural motifs in medicinal chemistry. This method also provides a new application of the Mitsunobu reaction.
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页码：157 / 162
页数：5
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