Synthesis of ivermectin-4″,5-diyl[bis(N-methylcarbamate)]

被引：0
|
作者：
A. N. Blinnikov
E. I. Chernoburova
N. G. Kolotyrkina
M. A. Shchetinina
V. A. Lishchuk
K. L. Ovchinnikov
A. V. Kolobov
M. Kh. Dzhafarov
F. I. Vasilevich
I. V. Zavarzin
机构：
[1] Russian Academy of Sciences,N. D. Zelinsky Institute of Organic Chemistry
[2] K. I. Skryabin Moscow State Academy of Veterinary Medicine and Biotechnology,undefined
来源：
Russian Chemical Bulletin | 2018年 / 67卷
关键词：
avermectin B; ivermectin; methyl isocyanate; MoO; Cl; (DMF); catalyst; ivermectin-4″,5-diyl[bis(; -methylcarbamate)]; antiparasitic activity;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
New ivermectin-4″,5-diyl[bis(N-methylcarbamate)] was synthesized by the MoO2Cl2(DMF)2-catalyzed reaction of ivermectin with methyl isocyanate. The synthesized compound could find application as antiparasitic agent.
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页码：833 / 835
页数：2
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