Interaction of aminoquinolines with unsaturated carboxylic acids. 1. Synthesis of N-quinolyl-β-alanines and their biological activity

被引：0
|
作者：
Beresnevicius Z.J. [1 ]
Viliunas V. [1 ]
Kantminiene K. [1 ]
机构：
[1] Kaunas University of Technology
来源：
Chemistry of Heterocyclic Compounds | 2000年 / 36卷 / 04期
关键词：
Aminoquinolines; Biological activity; Hydrazides; N-quinolyl-β-alanines;
D O I：
10.1007/BF02269541
中图分类号：
学科分类号：
摘要：
N-Quinolyl-β-alanines, and α-methyl- and β-methyl-N-quinolyl-β-alanines were prepared by reaction of aminoquinolines and acrylic, methacrylic, and crotonic acids. The corresponding hydrazides and benzylidenehydrazides were obtained. 4-Aminoquinoline with unsaturated acids in water gave betaines. The biological activity of sodium salts of β-alanines was investigated.
引用
收藏
页码：432 / 438
页数：6
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