Cyclocondensations of 3-alkylpyrazol-5-amines with 3-arylprop-2-enals and cyclic 1,3-diketones

被引：0

作者：

N. I. Zemlyanaya

V. V. Borodina

V. I. Musatov

S. V. Shishkina

D. S. Sofronov

V. V. Lipson

机构：

[1] National Academy of Medical Sciences of Ukraine,Danilevskii Institute of Endocrinous Pathology Problems

[2] National Academy of Sciences of Ukraine,Institute for Single Crystals

[3] Karazin Kharkiv National University,undefined

来源：

Russian Journal of Organic Chemistry | 2017年 / 53卷

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摘要：

Domino reactions of 3-alkylpyrazol-5-amines with 3-arylprop-2-enals and cyclic 1,3-diketones regioselectively afforded pyrazolo[3,4-b]pyridine derivatives. The alkylation and acylation of the synthesized compounds were studied using 3,7,7-trimethyl-4-[(E)-2-phenylethenyl]-2,4,6,7,8,9-hexahydro-5H-pyrazolo-[3,4-b]quinolin-5-one as model.

引用

页码：582 / 591

页数：9

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