Assessment of 18F-labeled mitochondrial complex I inhibitors as PET myocardial perfusion imaging agents in rats, rabbits, and primates

被引:0
|
作者
Ming Yu
Mary Guaraldi
Mikhail Kagan
Mahesh Mistry
Jennifer McDonald
Jody Bozek
Padmaja Yalamanchili
Megan Hayes
Michael Azure
Ajay Purohit
Heike Radeke
David S. Casebier
Simon P. Robinson
机构
[1] Bristol Myers Squibb Medical Imaging,Discovery Biology
[2] Bristol Myers Squibb Medical Imaging,Discovery Chemistry
关键词
Mitochondrial complex I Inhibitor; F; Cardiac PET; Myocardial perfusion imaging;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:63 / 72
页数:9
相关论文
共 50 条
  • [11] Stratification of 18F-Labeled PET Imaging Agents for the Assessment of Antiangiogenic Therapy Responses in Tumors
    Goggi, Julian L.
    Bejot, Romain
    Moonshi, Shehzahdi S.
    Bhakoo, Kishore K.
    JOURNAL OF NUCLEAR MEDICINE, 2013, 54 (09) : 1630 - 1636
  • [12] Synthesis of 18F-labeled acridinium cations: a new class of potential myocardial perfusion imaging agents.
    Inkster, James
    Dearling, Jason
    Snay, Erin
    Packard, Alan
    JOURNAL OF NUCLEAR MEDICINE, 2019, 60
  • [13] Initial characterization of an 18F-labeled myocardial perfusion tracer
    Huisman, Marc C.
    Higuchi, Takahiro
    Reder, Sybille
    Nekolla, Stephan G.
    Poethko, Thorsten
    Wester, Hans-Juergen
    Ziegler, Sibylle I.
    Casebier, David S.
    Robinson, Simon P.
    Schwaiger, Markus
    JOURNAL OF NUCLEAR MEDICINE, 2008, 49 (04) : 630 - 636
  • [14] Construction and Preliminary Evaluation of Two 18F-Labeled Radiopharmaceuticals for Myocardial Perfusion Imaging
    Lu, Xinmiao
    Deng, Xiaohui
    Kong, Fei
    Hai, Wangxi
    Luo, Quanyong
    ANALYTICAL CHEMISTRY, 2024, 96 (29) : 11725 - 11733
  • [15] Comparison of 18F-Labeled Fluoroalkylphosphonium Cations with 13N-NH3 for PET Myocardial Perfusion Imaging
    Kim, Dong-Yeon
    Kim, Hyeon Sik
    Reder, Sybille
    Zheng, Jin Hai
    Herz, Michael
    Higuchi, Takahiro
    Pyo, AYoung
    Bom, Hee-Seung
    Schwaiger, Markus
    Min, Jung-Joon
    JOURNAL OF NUCLEAR MEDICINE, 2015, 56 (10) : 1581 - 1586
  • [16] Evaluation of 18F-labeled icotinib derivatives as potential PET agents for tumor imaging
    Ren, Hongyu
    Ning, Hongyu
    Chang, Jin
    Zhao, Mingxia
    He, Yong
    Chong, Yan
    Qi, Chuanmin
    JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY, 2016, 309 (02) : 517 - 523
  • [17] Evaluation of 18F-labeled icotinib derivatives as potential PET agents for tumor imaging
    Hongyu Ren
    Hongyu Ning
    Jin Chang
    Mingxia Zhao
    Yong He
    Yan Chong
    Chuanmin Qi
    Journal of Radioanalytical and Nuclear Chemistry, 2016, 309 : 517 - 523
  • [18] Advances in PET myocardial perfusion imaging: F-18 labeled tracers
    Christoph Rischpler
    Min-Jae Park
    George S. K. Fung
    Mehrbod Javadi
    Benjamin M. W. Tsui
    Takahiro Higuchi
    Annals of Nuclear Medicine, 2012, 26 : 1 - 6
  • [19] F-18-labeled rhodamines as PET tracers for myocardial perfusion imaging
    Zhang, S.
    Bartholomae, M.
    Treves, S. T.
    Packard, A. B.
    JOURNAL OF NUCLEAR MEDICINE, 2012, 53 (04) : 671 - 671
  • [20] Advances in PET myocardial perfusion imaging: F-18 labeled tracers
    Rischpler, Christoph
    Park, Min-Jae
    Fung, George S. K.
    Javadi, Mehrbod
    Tsui, Benjamin M. W.
    Higuchi, Takahiro
    ANNALS OF NUCLEAR MEDICINE, 2012, 26 (01) : 1 - 6