Selective ligands of estrogen receptor β discovered using pharmacophore mapping and structure-based virtual screening

被引：0
|
作者：
Lei Chen
Dang Wu
Han-ping Bian
Guang-lin Kuang
Jing Jiang
Wei-hua Li
Gui-xia Liu
Shi-en Zou
Jin Huang
Yun Tang
机构：
[1] Shanghai Key Laboratory of New Drug Design,Department of Gynecology
[2] School of Pharmacy,undefined
[3] East China University of Science and Technology,undefined
[4] Obstetrics and Gynecology Hospital,undefined
[5] Fudan University,undefined
来源：
Acta Pharmacologica Sinica | 2014年 / 35卷
关键词：
estrogen receptor; subtype-selective ligand; estradiol; tamoxifen; pharmacophore mapping; structure-based virtual screening; breast cancer; anti-proliferation; cell cycle arrest;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
引用
收藏
页码：1333 / 1341
页数：8
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