Tetra-substituted pyrazole analogues: synthesis, molecular docking, ADMET prediction, antioxidant and pancreatic lipase inhibitory activities

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作者
Adnan Cetin
Ali Donmez
Abdullah Dalar
Ishak Bildirici
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[1] Van Yuzuncu Yil University,Department of Chemistry, Faculty of Education
[2] Van Yuzuncu Yil University,Department of Pharmaceutical Chemistry, Faculty of Pharmacy
[3] Van Yuzuncu Yil University,Department of Pharmaceutical Botany, Faculty of Pharmacy
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摘要
Synthesis, characterization and biological properties of tetra-substituted pyrazole analogues.Discovery of tetra-substituted pyrazole analogues as potential Pancreatic lipase enzyme inhibitor.Molecular docking studies of the tetra-substituted pyrazole analogues.A molecular approach in drug development for obesity disease.
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页码:189 / 204
页数:15
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