Synthesis of imidazo[1,2-a]pyrazine and imidazo[1,2-a]pyrimidine derivatives

被引：0

作者：

A. V. Borisov

A. A. Tolmachev

O. A. Zavada

I. A. Zhuravel’

S. N. Kovalenko

机构：

[1] Enamine Ltd,Institute of Organic Chemistry

[2] National Academy of Sciences of Ukraine,undefined

[3] National University of Pharmacy,undefined

来源：

Chemistry of Heterocyclic Compounds | 2013年 / 49卷

关键词：

2-aminoimidazole; imidazo[1,2-; ]pyrazines; imidazo[1,2-; ]pyrimidines; catalytic hydro-genation;

D O I：

暂无

中图分类号：

学科分类号：

摘要：

Synthetic approaches to the construction of bicyclic systems containing the imidazole nucleus have been considered. Methods for obtaining derivatives of imidazo[1,2-a]pyrazine and imidazo[1,2-a]pyrimidine have been studied, and methods have been developed for catalytic hydrogenation of these compounds. Partial reduction of the imidazole ring on imidazo[1,2-a]pyrimidine hydrogenation has been discovered for the first time.

引用

页码：704 / 711

页数：7

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