Design, radio-synthesis and evaluation of a novel [18F]-TKP for noninvasive PET imaging of brain Aβ deposits and neurofibrillary tangles

被引:0
|
作者
Kong, Yanyan [2 ]
Hua, Fengchun [2 ]
Guan, Yihui [2 ]
Zhao, Bizeng [1 ]
机构
[1] Jiaotong Univ, Shanghai Peoples Hosp 6, Shanghai, Peoples R China
[2] Fudan Univ, Huashan Hosp, PET Ctr, Shanghai, Peoples R China
基金
中国国家自然科学基金;
关键词
D O I
暂无
中图分类号
R8 [特种医学]; R445 [影像诊断学];
学科分类号
1002 ; 100207 ; 1009 ;
摘要
1030
引用
收藏
页数:2
相关论文
共 50 条
  • [41] Evaluation of [18F]-CP18 as a PET Imaging Tracer for Apoptosis
    Su, Helen
    Chen, Gang
    Gangadharmath, Umesh
    Gomez, Luis F.
    Liang, Qianwa
    Mu, Fanrong
    Mocharla, Vani P.
    Szardenings, A. Katrin
    Walsh, Joseph C.
    Xia, Chun-Fang
    Yu, Chul
    Kolb, Hartmuth C.
    MOLECULAR IMAGING AND BIOLOGY, 2013, 15 (06) : 739 - 747
  • [42] Evaluation of [18F]-CP18 as a PET Imaging Tracer for Apoptosis
    Helen Su
    Gang Chen
    Umesh Gangadharmath
    Luis F. Gomez
    Qianwa Liang
    Fanrong Mu
    Vani P. Mocharla
    A Katrin Szardenings
    Joseph C. Walsh
    Chun-Fang Xia
    Chul Yu
    Hartmuth C. Kolb
    Molecular Imaging and Biology, 2013, 15 : 739 - 747
  • [43] Radiosynthesis and Preclinical Evaluation of m-[18F]FET and [18F]FET-OMe as Novel [18F]FET Analogs for Brain Tumor Imaging
    Groener, Benedikt
    Hoffmann, Chris
    Endepols, Heike
    Urusova, Elizaveta A.
    Brugger, Melanie
    Neumaier, Felix
    Timmer, Marco
    Neumaier, Bernd
    Zlatopolskiy, Boris D.
    MOLECULAR PHARMACEUTICS, 2024, 21 (06) : 2795 - 2812
  • [44] PET IMAGING OF [18F]DOTK8-SFB: A NOVEL 18F BASED RADIOTRACER FOR IMAGING OF OXYTOCIN RECEPTORS
    Parmar, A.
    Pascali, G.
    Hering, A.
    Rahardjo, G.
    Arthur, A.
    Hamze, H.
    Zahra, D.
    Zhang, B.
    McKay, T.
    Markham, J.
    Matesic, L.
    Klenner, M. A.
    Tran, M.
    Banati, R.
    Gregoire, M. C.
    Muttenthaler, M.
    Guastella, A. J.
    INTERNAL MEDICINE JOURNAL, 2021, 51 : 9 - 9
  • [45] Synthesis and Biological Evaluation of [18F]FECNT-d4 as a Novel PET Agent for Dopamine Transporter Imaging
    Shanshan Cao
    Jie Tang
    Chunyi Liu
    Yi Fang
    Linyang Ji
    Yingjiao Xu
    Zhengping Chen
    Molecular Imaging and Biology, 2021, 23 : 733 - 744
  • [46] Synthesis and Biological Evaluation of [18F]FECNT-d4 as a Novel PET Agent for Dopamine Transporter Imaging
    Cao, Shanshan
    Tang, Jie
    Liu, Chunyi
    Fang, Yi
    Ji, Linyang
    Xu, Yingjiao
    Chen, Zhengping
    MOLECULAR IMAGING AND BIOLOGY, 2021, 23 (05) : 733 - 744
  • [47] Radiosynthesis and preclinical evaluation of [18F]FEM as a potential novel PET probe for tumor imaging
    Jiang, Yanping
    Zhou, Wenlan
    Hu, Kongzhen
    Han, Yanjiang
    Sun, Penghui
    Wang, Quanshi
    Li, Guiping
    Wu, Hubing
    Tang, Ganghua
    Huang, Shun
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 30 (12)
  • [48] Automated Radiolabeling and Evaluation of [18F]FPMBBG: A Novel Cardiac Neuronal PET Imaging Agent
    Ju, Min
    Ren, Wanjie
    Zhang, Zongyao
    Lu, Jie
    Han, Kai
    Wang, Lei
    Fang, Wei
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2025, 68 (03):
  • [49] Preclinical evaluation of [18F]SYN1 and [18F]SYN2, novel radiotracers for PET myocardial perfusion imaging
    Krajewski, Seweryn
    Steczek, Lukasz
    Gotowicz, Karina
    Karczmarczyk, Urszula
    Towpik, Joanna
    Witkowska-Patena, Ewa
    Lyczko, Krzysztof
    Mazur, Maciej
    Kozanecki, Przemyslaw
    Wlostowska, Joanna
    Knuuti, Juhani
    Dziuk, Miroslaw
    Garnuszek, Piotr
    Kozanecki, Cezary
    EJNMMI RESEARCH, 2024, 14 (01):
  • [50] A novel approach to the synthesis of [18F]flumazenil, a radioligand for PET imaging of central benzodiazepine receptors
    M. Nasirzadeh
    D. D. Vaulina
    O. F. Kuznetsova
    N. A. Gomzina
    Russian Chemical Bulletin, 2016, 65 : 794 - 800