Synthesis of 5,4"-di-O-succinoylavermectin B1

被引：12

作者：

Chernoburova, E. I. ^{[1
]}

Danchenko, K. V. ^{[1
]}

Shchetinina, M. A. ^{[1
]}

Zharov, A. A. ^{[1
]}

Kolobov, A. V. ^{[2
]}

Dzhafarov, M. Kh. ^{[3
]}

Vasilevich, F. I. ^{[3
]}

Zavarzin, I. V. ^{[1
]}

机构：

[1] Russian Acad Sci, ND Zelinsky Inst Organ Chem, 47 Leninsky Prosp, Moscow 119991, Russia

[2] Yaroslavl State Tech Univ, 88 Moskovskii Prosp, Yaroslavl 150023, Russia

[3] KI Skryabin Moscow State Acad Vet Med & Biotechno, 23 Ul Akad Skryabina, Moscow 119991, Russia

来源：

RUSSIAN CHEMICAL BULLETIN | 2016年 / 65卷 / 12期

基金：

俄罗斯科学基金会;

关键词：

ultrahigh pressure; avermectin B-1; succinic anhydride; 5,4 ''-di-O-succinoylavermectin B-1; acylation reaction; antiparasitic activity; IVERMECTIN; PARASITES; TOXICITY;

D O I：

10.1007/s11172-016-1684-5

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A reaction of avermectin B-1 with succinic anhydride at ultrahigh pressure (10 kbar) gave previously unavailable 5,4"-di-O-succinoylavermectin B-1, which is of interest as potential antiparasitic agent.

引用

页码：2952 / 2955

页数：4

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