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- [11] Flavokawain A is a natural inhibitor of PRMT5 in bladder cancerJournal of Experimental & Clinical Cancer Research, 41Shuangjie Liu论文数: 0 引用数: 0 h-index: 0机构: The First Hospital of China Medical University,Department of UrologyZhuonan Liu论文数: 0 引用数: 0 h-index: 0机构: The First Hospital of China Medical University,Department of UrologyChiyuan Piao论文数: 0 引用数: 0 h-index: 0机构: The First Hospital of China Medical University,Department of UrologyZhe Zhang论文数: 0 引用数: 0 h-index: 0机构: The First Hospital of China Medical University,Department of UrologyChuize Kong论文数: 0 引用数: 0 h-index: 0机构: The First Hospital of China Medical University,Department of UrologyLei Yin论文数: 0 引用数: 0 h-index: 0机构: The First Hospital of China Medical University,Department of UrologyXi Liu论文数: 0 引用数: 0 h-index: 0机构: The First Hospital of China Medical University,Department of Urology
- [12] Discovery of novel potent and selective inhibitors of PRMT5 with anti-tumor activity in hepatocellular carcinoma and lung pre-clinical modelsCANCER RESEARCH, 2020, 80 (16)Gonzalvez, Francois论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, Leuven, Belgium Aligos Therapeut, Leuven, BelgiumVandyck, Koen论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, Leuven, Belgium Aligos Therapeut, Leuven, BelgiumDebing, Yannick论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, Leuven, Belgium Aligos Therapeut, Leuven, BelgiumGupta, Kusum论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, San Francisco, CA USA Aligos Therapeut, Leuven, BelgiumMisner, Dinah论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, San Francisco, CA USA Aligos Therapeut, Leuven, BelgiumZhang, Qingling论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, San Francisco, CA USA Aligos Therapeut, Leuven, BelgiumLiu, Jyanwei论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, San Francisco, CA USA Aligos Therapeut, Leuven, BelgiumStoycheva, Antitsa论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, San Francisco, CA USA Aligos Therapeut, Leuven, BelgiumStevens, Sarah论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, San Francisco, CA USA Aligos Therapeut, Leuven, BelgiumSymons, Julian论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, San Francisco, CA USA Aligos Therapeut, Leuven, BelgiumBeigelman, Leonid论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, San Francisco, CA USA Aligos Therapeut, Leuven, BelgiumRaboisson, Pierre论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, Leuven, Belgium Aligos Therapeut, Leuven, BelgiumDeval, Jerome论文数: 0 引用数: 0 h-index: 0机构: Aligos Therapeut, San Francisco, CA USA Aligos Therapeut, Leuven, Belgium
- [13] PRMT5, a Novel Epigenetic Target in Lung CancersEUROPEAN JOURNAL OF CANCER, 2012, 48 : 171 - 171Otterson, G. A.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USA Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USAWu, X.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USA Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USAWelliver, M.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Radiat Oncol, Columbus, OH 43210 USA Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USASharma, S.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Radiat Oncol, Columbus, OH 43210 USA Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USAShilo, K.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Pathol, Columbus, OH 43210 USA Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USAHitchcock, C.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Pathol, Columbus, OH 43210 USA Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USALi, C.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USABaiocchi, R.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Columbus, OH 43210 USA Ohio State Univ, Div Med Oncol, Columbus, OH 43210 USA
- [14] DISCOVERY AND PHARMACOLOGICAL CHARACTERIZATION OF SKL27969, A NOVEL BRAINPENETRATING PRMT5 INHIBITOR WITH STRONG ANTITUMOR ACTIVITY, IN GLIOBLASTOMA AND BRAIN METASTASIS PRECLINICAL MODELSNEURO-ONCOLOGY, 2022, 24 : 233 - 234Moon, Mijin论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut Co Ltd, Seongnam, South Korea SK Biopharmaceut Co Ltd, Seongnam, South KoreaShin, Yongje论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut Co Ltd, Seongnam, South Korea SK Biopharmaceut Co Ltd, Seongnam, South KoreaLee, Ho Yeon论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut Co Ltd, Seongnam, South Korea SK Biopharmaceut Co Ltd, Seongnam, South KoreaHong, Beomjin论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut Co Ltd, Seongnam, South Korea SK Biopharmaceut Co Ltd, Seongnam, South KoreaKim, Jinhee论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut Co Ltd, Seongnam, South Korea SK Biopharmaceut Co Ltd, Seongnam, South KoreaLee, Jun论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut Co Ltd, Seongnam, South Korea SK Biopharmaceut Co Ltd, Seongnam, South KoreaLaramy, Janice K.论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Inc, Paramus, NJ USA SK Biopharmaceut Co Ltd, Seongnam, South KoreaVashi, Vijaykumar论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Inc, Paramus, NJ USA SK Biopharmaceut Co Ltd, Seongnam, South KoreaPark, Sook-Kyung论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut Co Ltd, Seongnam, South Korea SK Biopharmaceut Co Ltd, Seongnam, South Korea
- [15] Discovery and In Vivo Efficacy of AZ-PRMT5i-1, a Novel PRMT5 Inhibitor with High MTA CooperativityJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (16) : 13604 - 13638Smith, James M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandBarlaam, Bernard论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandBeattie, David论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandBradshaw, Lauren论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandChan, Ho Man论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandChiarparin, Elisabetta论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandCollingwood, Olga论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandCooke, Sophie L.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandCronin, Anna论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandCumming, Iain论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandDean, Emma论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandDebreczeni, Judit E.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, Englanddel Barco Barrantes, Ivan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandDiene, Coura论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandGianni, Davide论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandGuerot, Carine论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandGuo, Xiaoxiao论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandGuven, Sinem论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandHayhow, Thomas G.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandHong, Ted论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandKemmitt, Paul D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandLamont, Gillian M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandLamont, Scott论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandLynch, James T.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandMcWilliams, Lisa论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandMoore, Shaun论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandRaubo, Piotr论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandRobb, Graeme R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandRobinson, James论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandScott, James S.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandSrinivasan, Bharath论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandSteward, Oliver论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandStubbs, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandSyson, Karl论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandTan, Lixiang论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, Beijing 100176, Peoples R China AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandTurner, Oliver论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandUnderwood, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandUrosevic, Jelena论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandVazquez-Chantada, Mercedes论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandWhittaker, Amy L.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandWilson, David M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandWinter-Holt, Jon J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England
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- [17] PRMT5 Selective Inhibitor Enhances Therapeutic Efficacy of Cisplatin in Lung Cancer CellsINTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2021, 22 (11)论文数: 引用数: h-index:机构:Ramakrishnan, Rakhee K.论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates Univ Sharjah, Sharjah Inst Med Res, Sharjah 27272, U Arab Emirates Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates论文数: 引用数: h-index:机构:Omar, Hany A.论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Sharjah Inst Med Res, Sharjah 27272, U Arab Emirates Univ Sharjah, Coll Pharm, Sharjah 27272, U Arab Emirates Univ Sharjah, Coll Med, Sharjah 27272, U Arab EmiratesSaheb Sharif-Askari, Narjes论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates Univ Sharjah, Sharjah Inst Med Res, Sharjah 27272, U Arab Emirates Univ Sharjah, Coll Med, Sharjah 27272, U Arab EmiratesShafarin, Jasmin论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Sharjah Inst Med Res, Sharjah 27272, U Arab Emirates Univ Sharjah, Coll Med, Sharjah 27272, U Arab EmiratesElmoselhi, Adel B.论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates Michigan State Univ, Dept Physiol, E Lansing, MI 48824 USA Univ Sharjah, Coll Med, Sharjah 27272, U Arab EmiratesIhmaid, Ahmed论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates Univ Sharjah, Coll Med, Sharjah 27272, U Arab EmiratesAlHaj Ali, Suhib论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates Univ Sharjah, Coll Med, Sharjah 27272, U Arab EmiratesAlalool, Abdulla论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates Univ Sharjah, Coll Med, Sharjah 27272, U Arab EmiratesAbdullah, Reem论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates Univ Sharjah, Coll Med, Sharjah 27272, U Arab EmiratesHamid, Qutayba论文数: 0 引用数: 0 h-index: 0机构: Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates Univ Sharjah, Sharjah Inst Med Res, Sharjah 27272, U Arab Emirates McGill Univ, Ctr Hlth, Meakins Christie Labs, Res Inst, Montreal, PQ H4A 3J1, Canada Univ Sharjah, Coll Med, Sharjah 27272, U Arab Emirates
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