Discovery of TRV130, a G protein biased agonist of the μ-opioid receptor, for the treatment of acute severe pain

被引:0
|
作者
Crombie, Aimee [1 ]
Chen, Xiao-Tao [1 ]
Pitis, Philip [1 ]
Liu, Guodong [1 ]
Yuan, Catherine [1 ]
Gotchev, Dimitar [4 ]
Yamashita, Dennis [3 ]
Violin, Jonathan [2 ]
机构
[1] Trevena Inc, Chem, King Of Prussia, PA USA
[2] Trevena Inc, Biol, King Of Prussia, PA USA
[3] GSK, Discovery Partnerships Acad, Boston, PA USA
[4] Teva Pharmaceut, Chem, W Chester, PA USA
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O6 [化学];
学科分类号
0703 ;
摘要
34
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页数:2
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