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- [21] Discovery of SHR9352: A Highly Potent G Protein-Biased μ-Opioid Receptor Agonist ACS OMEGA, 2017, 2 (12): : 9261 - 9267
- [22] APOLLO-1: Phase 3 Study of Oliceridine (TRV130) for Management of Acute Pain ANESTHESIA AND ANALGESIA, 2017, 124 : 744 - 744
- [23] Structure Activity Relationships and Discovery of a G Protein Biased μ Opioid Receptor Ligand, [(3-Methoxythiophen-2-yl)methyl]a2[(9R)-9-(pyridin-2-y1)-6-oxaspiro-[4.5]clecan-9-yl]ethylpamine (TRV130), for the Treatment of Acute Severe Pain JOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (20) : 8019 - 8031
- [24] Desmetramadol Is Identified as a G-Protein Biased μ Opioid Receptor Agonist FRONTIERS IN PHARMACOLOGY, 2020, 10
- [25] TRV130, a novel biased opioid ligand, elicits increased analgesia with reduced adverse effects compared to morphine in healthy volunteers JOURNAL OF PAIN, 2014, 15 (04): : S95 - S95
- [26] A Novel G Protein-Biased Agonist at the δ Opioid Receptor with Analgesic Efficacy in Models of Chronic Pain JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2020, 372 (02): : 224 - 236
- [28] TRV0109101, a G Protein-Biased Agonist of the μ-Opioid Receptor, Does Not Promote Opioid-Induced Mechanical Allodynia following Chronic Administration JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2017, 362 (02): : 254 - 262
- [30] Can oliceridine (TRV130), an ideal novel. receptor G protein pathway selective (μ-GPS) modulator, provide analgesia without opioid-related adverse reactions? KOREAN JOURNAL OF PAIN, 2018, 31 (02): : 73 - 79