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- [1] Design of potent and selective human cathepsin K inhibitors that span the active sitePROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1997, 94 (26) : 14249 - 14254Thompson, SK论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAHalbert, SM论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USABossard, MJ论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USATomaszek, TA论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USALevy, MA论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAZhao, BG论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USASmith, WW论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAAbdel-Meguid, SS论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAJanson, CA论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAD'Alessio, KJ论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAMcQueney, MS论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAAmegadzie, BY论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAHanning, CR论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USADesJarlais, RL论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USABriand, J论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USASarkar, SK论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAHuddleston, MJ论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAIjames, CF论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USACarr, SA论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAGarnes, KT论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAShu, A论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAHeys, JR论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USABradbeer, J论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAZembryki, D论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USALee-Rykaczewski, L论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAJames, IE论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USALark, MW论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USADrake, FH论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAGowen, M论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAGleason, JG论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USAVeber, DF论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USA
- [2] Structure and design of potent and selective cathepsin K inhibitorsJOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1997, 119 (46) : 11351 - 11352Yamashita, DS论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Smith, WW论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Zhao, BG论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Janson, CA论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Tomaszek, TA论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Bossard, MJ论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Levy, MA论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Oh, HJ论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Carr, TJ论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Thompson, SK论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Ijames, CF论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Carr, SA论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406McQueney, M论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406DAlessio, KJ论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Amegadzie, BY论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Hanning, CR论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406AbdelMeguid, S论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406DesJarlais, RL论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Gleason, JG论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406Veber, DF论文数: 0 引用数: 0 h-index: 0机构: SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406
- [3] Potent and selective cathepsin K inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY, 2006, 14 (20) : 6789 - 6806Shinozuka, Tsuyoshi论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanShimada, Kousei论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanMatsui, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanYamane, Takahiro论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanAma, Mayumi论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanFukuda, Takeshi论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanTaki, Motohiko论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanTakeda, Yuko论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanOtsuka, Eri论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanYamato, Michiko论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanMochizuki, Shin-ichi论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanOhhata, Keiko论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, JapanNaito, Satoru论文数: 0 引用数: 0 h-index: 0机构: Sankyo Co Ltd, Med Chem Res Labs, Shinagawa Ku, Tokyo 1408710, Japan
- [4] Thiosemicarbazones as potent and selective cathepsin K inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 241Chavarria, Gustavo E.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USADevanna, Kishore K. Gaddale论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAJones, Lindsay M.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAMacDonough, Matthew T.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAYoo, Grace K.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USALocke, Ashleigh论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USADeliz, Rafael论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAChaplin, David J.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USASiim, Bronwyn G.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAChen, Shen-En论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAPinney, Kevin G.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USATrawick, Mary L.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA
- [5] Design of potent, selective, and orally bioavailable inhibitors of cysteine protease cathepsin KJOURNAL OF MEDICINAL CHEMISTRY, 2004, 47 (03) : 588 - 599Tavares, FX论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USA GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USABoncek, V论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USADeaton, DN论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USAHassell, AM论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USALong, ST论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USAMiller, AB论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USAPayne, AA论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USAMiller, LR论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USAShewchuk, LM论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USAWells-Knecht, K论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USAWillard, DH论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USAWright, LL论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USAZhou, HQ论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Med Chem, Res Triangle Pk, NC USA
- [6] Design and synthesis of potent and selective inhibitors of the osteoclast-specific cysteine protease, cathepsin KPEPTIDE SCIENCE - PRESENT AND FUTURE, 1999, : 628 - 630Veber, DF论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAMarquis, RW论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USARu, Y论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAYamashita, DS论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAOh, HJ论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAThompson, SK论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAHalbert, SM论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USACarr, TJ论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAGleason, JG论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USATomaszek, TA论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USALevy, MA论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USABossard, M论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USATew, DG论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAJames, IE论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USABriand, J论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USACarr, SA论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAZymbryki, D论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USALee-Rykaczewski, L论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USADesjarlais, RL论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAMcQueney, MS论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAD'Alessio, KJ论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAZhao, B论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAJanson, CA论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USAAbdel-Meguid, SS论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USASmith, WW论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA SmithKline Beecham Pharmaceut, King Of Prussia, PA 19406 USA
- [7] Rational design of potent and selective NH-linked aryl/heteroaryl cathepsin K inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (16) : 4291 - 4295Robichaud, J论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3L1, CanadaBayly, C论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3L1, CanadaOballa, R论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3L1, CanadaPrasit, P论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3L1, CanadaMellon, C论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3L1, CanadaFalgueyret, JP论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3L1, CanadaPercival, MD论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3L1, CanadaWesolowski, G论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3L1, CanadaRodan, SB论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3L1, Canada
- [8] The use of selective inhibitors for computer modeling of monoamine oxidases active site.VOPROSY MEDITSINSKOI KHIMII, 1997, 43 (06): : 527 - 536Veselovsky, AV论文数: 0 引用数: 0 h-index: 0机构: Inst Biomed Chem, Moscow 119832, Russia Inst Biomed Chem, Moscow 119832, RussiaIvanov, AS论文数: 0 引用数: 0 h-index: 0机构: Inst Biomed Chem, Moscow 119832, Russia Inst Biomed Chem, Moscow 119832, RussiaMedvedev, AE论文数: 0 引用数: 0 h-index: 0机构: Inst Biomed Chem, Moscow 119832, Russia Inst Biomed Chem, Moscow 119832, Russia
- [9] The consequences of lysosomotropism on the design of selective cathepsin K inhibitorsCHEMBIOCHEM, 2006, 7 (10) : 1525 - 1535Black, W. Cameron论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem & Biochem, Pointe Claire, PQ H9R 4P8, CanadaPercival, M. David论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Dept Med Chem & Biochem, Pointe Claire, PQ H9R 4P8, Canada
- [10] Cathepsin K and the design of inhibitors of cathepsin KCURRENT PHARMACEUTICAL DESIGN, 2000, 6 (01) : 1 - 24Yamashita, DS论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USADodds, RA论文数: 0 引用数: 0 h-index: 0机构: SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USA