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- [41] Phase 1 study of single-agent WNT974, a first-in-class Porcupine inhibitor, in patients with advanced solid tumoursBRITISH JOURNAL OF CANCER, 2021, 125 (01) : 28 - 37Rodon, Jordi论文数: 0 引用数: 0 h-index: 0机构: Vall dHebron Univ Hosp, Barcelona, Spain Univ Autonoma Barcelona, Barcelona, Spain Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Vall dHebron Univ Hosp, Barcelona, SpainArgiles, Guillem论文数: 0 引用数: 0 h-index: 0机构: Vall dHebron Univ Hosp, Barcelona, Spain Univ Autonoma Barcelona, Barcelona, Spain Vall dHebron Univ Hosp, Barcelona, SpainConnolly, Roisin M.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sch Med, Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Univ Coll Cork, Coll Med & Hlth, CancerRes UCC, Cork, Ireland Vall dHebron Univ Hosp, Barcelona, SpainVaishampayan, Ulka论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Dept Oncol, Karmanos Canc Inst, Detroit, MI USA Vall dHebron Univ Hosp, Barcelona, Spainde Jonge, Maja论文数: 0 引用数: 0 h-index: 0机构: Erasmus MC, Dept Med Oncol, Canc Inst, Rotterdam, Netherlands Vall dHebron Univ Hosp, Barcelona, SpainGarralda, Elena论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ Madrid Sanchinarro, START Madrid, Madrid, Spain Vall dHebron Univ Hosp, Barcelona, Spain论文数: 引用数: h-index:机构:Smith, David C.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ann Arbor, MI 48109 USA Vall dHebron Univ Hosp, Barcelona, SpainDobson, Jason R.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Cambridge, MA USA Vall dHebron Univ Hosp, Barcelona, SpainMcLaughlin, Margaret E.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Cambridge, MA USA Vall dHebron Univ Hosp, Barcelona, SpainSeroutou, Abdelkader论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Basel, Switzerland Vall dHebron Univ Hosp, Barcelona, SpainJi, Yan论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, E Hanover, NJ USA Vall dHebron Univ Hosp, Barcelona, SpainMorawiak, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Cambridge, MA USA Vall dHebron Univ Hosp, Barcelona, SpainMoody, Susan E.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Cambridge, MA USA Vall dHebron Univ Hosp, Barcelona, SpainJanku, Filip论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USA Vall dHebron Univ Hosp, Barcelona, Spain
- [42] A Phase 1 dose escalation study of TACH101, a first-in-class KDM4 inhibitor for advanced solid tumorsMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Tsimberidou, Apostolia论文数: 0 引用数: 0 h-index: 0Vandross, Andrae L.论文数: 0 引用数: 0 h-index: 0Sommerhalder, David论文数: 0 引用数: 0 h-index: 0Joseph, Charmaine论文数: 0 引用数: 0 h-index: 0Chandhasin, Chandtip论文数: 0 引用数: 0 h-index: 0Perabo, Frank论文数: 0 引用数: 0 h-index: 0Clarke, Michael F.论文数: 0 引用数: 0 h-index: 0
- [43] Phase 1 study of single-agent WNT974, a first-in-class Porcupine inhibitor, in patients with advanced solid tumoursBritish Journal of Cancer, 2021, 125 : 28 - 37Jordi Rodon论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyGuillem Argilés论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyRoisin M. Connolly论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyUlka Vaishampayan论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyMaja de Jonge论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyElena Garralda论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyMarios Giannakis论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyDavid C. Smith论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyJason R. Dobson论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyMargaret E. McLaughlin论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyAbdelkader Seroutou论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyYan Ji论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyJennifer Morawiak论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologySusan E. Moody论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical OncologyFilip Janku论文数: 0 引用数: 0 h-index: 0机构: Vall d’Hebron University Hospital and Universitat Autònoma de Barcelona,Department of Medical Oncology
- [44] Phase 1 extension study of BBI503, a first-in-class cancer stemness kinase inhibitor, in patients with advanced colorectal cancerJOURNAL OF CLINICAL ONCOLOGY, 2015, 33 (15)Jonker, Derek J.论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaLaurie, Scott Andrew论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaCote, Gregory Michael论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaFlaherty, Keith论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaFuchs, Charles S.论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaChugh, Rashmi论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaSmith, David C.论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaEdenfield, William Jeffery论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaConkling, Paul R.论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaMier, James Walter论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaGoodwin, Rachel Anne论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaKwak, Eunice Lee论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaAbrams, Thomas Adam论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaGoel, Rakesh论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaCleary, James M.论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaLi, Wei论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaLi, Youzhi论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaJemison, Jamileh论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaHitron, Matthew论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, CanadaLi, Chiang论文数: 0 引用数: 0 h-index: 0机构: Ottawa Hosp Canc Ctr, Ottawa, ON, Canada
- [45] First-In-Human, First-In-Class, Phase I Trial of the Fucosylation Inhibitor SGN-2FF in Patients with Advanced Solid TumorsONCOLOGIST, 2021, 26 (11): : 925 - +Do, Khanh T.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USAChow, Laura Quan Man论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Seattle Canc Care Alliance, Seattle, WA 98195 USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USAReckamp, Karen论文数: 0 引用数: 0 h-index: 0机构: City Hope Comprehens Canc Ctr, Duarte, CA USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USASanborn, Rachel E.论文数: 0 引用数: 0 h-index: 0机构: Earle A Chiles Res Inst, Prov Canc Inst, Portland, OR USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USABurris, Howard论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USARobert, Francisco论文数: 0 引用数: 0 h-index: 0机构: Univ Alabama Birmingham, Birmingham, AL USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USACamidge, D. Ross论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Ctr Canc, Aurora, CO USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USASteuer, Conor E.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Sch Med, Winship Canc Inst, Atlanta, GA 30322 USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USAStrickler, John H.论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Med Ctr, Durham, NC USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USAWeise, Amy论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USASpecht, Jennifer M.论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Seattle Canc Care Alliance, Seattle, WA 98195 USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USAGutierrez, Martin论文数: 0 引用数: 0 h-index: 0机构: Hackensack Univ, Med Ctr, Hackensack, NJ USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USAHaughney, Peter论文数: 0 引用数: 0 h-index: 0机构: Seagen Inc, Bothell, WA USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USAHengel, Shawna论文数: 0 引用数: 0 h-index: 0机构: Seagen Inc, Bothell, WA USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USADerleth, Christina Louise论文数: 0 引用数: 0 h-index: 0机构: Seagen Inc, Bothell, WA USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USAYap, Timothy A.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, 1515 Holcombe Blvd, Houston, TX 77030 USA Dana Farber Canc Inst, 450 Brookline Ave, Boston, MA 02115 USA
- [46] A First-in-Human Phase 1 Study of Oral LOXO-338, a Selective BCL2 Inhibitor, in Patients with Advanced Hematologic Malignancies (Trial in Progress)BLOOD, 2021, 138Alencar, Alvaro J.论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USA Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USARoeker, Lindsey E.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USAHoffman, Marc论文数: 0 引用数: 0 h-index: 0机构: Univ Kansas, Ctr Canc, Hematol Malignancies & Cellular Therapeut, Overland Pk, KS USA Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USAMurthy, Guru Subramanian Guru论文数: 0 引用数: 0 h-index: 0机构: Med Coll Wisconsin, Div Hematol Oncol, Milwaukee, WI 53226 USA Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USAPatel, Vishalkumar论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Stamford, CT USA Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USAKu, Nora C.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Stamford, CT USA Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USAPauff, James M.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Stamford, CT USA Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USAEyre, Toby A.论文数: 0 引用数: 0 h-index: 0机构: Oxford Univ Hosp NHS Fdn Trust, Churchill Canc Ctr, Oxford, England Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USAJurczak, Wojciech论文数: 0 引用数: 0 h-index: 0机构: Maria Sklodowska Curie Natl Res Inst Oncol, Krakow, Poland Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USALe Gouill, Steven论文数: 0 引用数: 0 h-index: 0机构: NeXT Univ Nantes, INSERM CRCINA Nantes Angers, CHU Nantes, Serv Hematol Clin, Nantes, France Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USA
- [47] A first-in-human phase 1 study of oral LOXO-338, a selective BCL2 inhibitor, in patients with advanced hematologic malignancies (trial in progress)CLINICAL LYMPHOMA MYELOMA & LEUKEMIA, 2022, 22 : S37 - S38Kumar, Shaji论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin Rochester, Dept Hematol, Rochester, MN USA Mayo Clin Rochester, Dept Hematol, Rochester, MN USAKapoor, Prashant论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Internal Med, Div Hematol, Rochester, MN USA Mayo Clin Rochester, Dept Hematol, Rochester, MN USAAlencar, Alvaro论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Miller Sch Med, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USA Mayo Clin Rochester, Dept Hematol, Rochester, MN USAMurthy, Guru Subramanian Guru论文数: 0 引用数: 0 h-index: 0机构: Med Coll Wisconsin, Div Hematol Oncol, Milwaukee, WI 53226 USA Mayo Clin Rochester, Dept Hematol, Rochester, MN USA论文数: 引用数: h-index:机构:Pagel, John论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Stamford, CT USA Mayo Clin Rochester, Dept Hematol, Rochester, MN USAPatel, Vishalkumar论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Stamford, CT USA Mayo Clin Rochester, Dept Hematol, Rochester, MN USAPauff, James论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Stamford, CT USA Mayo Clin Rochester, Dept Hematol, Rochester, MN USAZinzani, Pier Luigi论文数: 0 引用数: 0 h-index: 0机构: Univ Bologna, Inst Hematol Seragnoli, Bologna, Italy Mayo Clin Rochester, Dept Hematol, Rochester, MN USALe Gouill, Steven论文数: 0 引用数: 0 h-index: 0机构: Inst Curie Hosp, F-75248 Paris, France Mayo Clin Rochester, Dept Hematol, Rochester, MN USAMato, Anthony R.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mayo Clin Rochester, Dept Hematol, Rochester, MN USAJurczak, Wojciech论文数: 0 引用数: 0 h-index: 0机构: Maria Sklodowska Curie Natl Res Inst Oncol, Krakow, Poland Mayo Clin Rochester, Dept Hematol, Rochester, MN USARoeker, Lindsey E.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mayo Clin Rochester, Dept Hematol, Rochester, MN USA
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- [50] First-in-Class, First-in-Human Phase I Study of Selinexor, a Selective Inhibitor of Nuclear Export, in Patients With Advanced Solid TumorsJOURNAL OF CLINICAL ONCOLOGY, 2016, 34 (34) : 4142 - +Razak, Albiruni R. Abdul论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, Canada Princess Margaret Canc Ctr, Toronto, ON, CanadaMau-Soerensen, Morten论文数: 0 引用数: 0 h-index: 0机构: Rigshosp, Copenhagen, Denmark Princess Margaret Canc Ctr, Toronto, ON, CanadaGabrail, Nashat Y.论文数: 0 引用数: 0 h-index: 0机构: Gabrail Canc Inst, Canton, OH USA Princess Margaret Canc Ctr, Toronto, ON, CanadaGerecitano, John F.论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Mem Sloan Kettering Canc Ctr, New York, NY USA Princess Margaret Canc Ctr, Toronto, ON, CanadaShields, Anthony F.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Princess Margaret Canc Ctr, Toronto, ON, CanadaUnger, Thaddeus J.论文数: 0 引用数: 0 h-index: 0机构: Karyopharm Therapeut, Newton, MA USA Princess Margaret Canc Ctr, Toronto, ON, CanadaSaint-Martin, Jean R.论文数: 0 引用数: 0 h-index: 0机构: Karyopharm Therapeut, Newton, MA USA Princess Margaret Canc Ctr, Toronto, ON, CanadaCarlson, Robert论文数: 0 引用数: 0 h-index: 0机构: Karyopharm Therapeut, Newton, MA USA Princess Margaret Canc Ctr, Toronto, ON, CanadaLandesman, Yosef论文数: 0 引用数: 0 h-index: 0机构: Karyopharm Therapeut, Newton, MA USA Princess Margaret Canc Ctr, Toronto, ON, CanadaMcCauley, Dilara论文数: 0 引用数: 0 h-index: 0机构: Karyopharm Therapeut, Newton, MA USA Princess Margaret Canc Ctr, Toronto, ON, CanadaRashal, Tami论文数: 0 引用数: 0 h-index: 0机构: Karyopharm Therapeut, Newton, MA USA Princess Margaret Canc Ctr, Toronto, ON, CanadaLassen, Ulrik论文数: 0 引用数: 0 h-index: 0机构: Rigshosp, Copenhagen, Denmark Princess Margaret Canc Ctr, Toronto, ON, CanadaKim, Richard论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA Princess Margaret Canc Ctr, Toronto, ON, CanadaStayner, Lee-Anne论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, Canada Princess Margaret Canc Ctr, Toronto, ON, CanadaMirza, Mansoor R.论文数: 0 引用数: 0 h-index: 0机构: Karyopharm Therapeut, Newton, MA USA Princess Margaret Canc Ctr, Toronto, ON, CanadaKauffman, Michael论文数: 0 引用数: 0 h-index: 0机构: Karyopharm Therapeut, Newton, MA USA Princess Margaret Canc Ctr, Toronto, ON, CanadaShacham, Sharon论文数: 0 引用数: 0 h-index: 0机构: Karyopharm Therapeut, Newton, MA USA Princess Margaret Canc Ctr, Toronto, ON, CanadaMahipal, Amit论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA Princess Margaret Canc Ctr, Toronto, ON, Canada